SCHEMBL9871528

SCHEMBL9871528

COC(=O)/C=C/c1ccccc1C1C(C(=O)O)=C(C)NC(C)=C1C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 4/20 0.57
LMNA P02545 3/20 0.57
CYP2C9 P11712 3/20 0.57
CYP2C19 P33261 3/20 0.57
CYP3A4 P08684 2/20 0.57
TBXAS1 P24557 2/20 0.57
KCNH2 Q12809 2/20 0.57
HTT P42858 2/20 0.57
NR1I2 O75469 2/20 0.57
PGR P06401 1/20 0.57
SLC6A2 P23975 1/20 0.57
DRD3 P35462 1/20 0.57
OPRK1 P41145 1/20 0.57
PDE4D Q08499 1/20 0.57
CACNA1B Q00975 7/20 0.43
MAPT P10636 4/20 0.43
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 3/20 0.43
TP53 P04637 2/20 0.43
CYP1A2 P05177 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871535 1.00 ADORA3 (0.57) ADORA3LMNACYP2C9CYP2C19CYP3A4
SCHEMBL9871869 0.88 ADORA3 (0.67) ADORA3LMNACYP2C9CYP2C19CYP3A4
SCHEMBL9871872 0.88 ADORA3 (0.67) ADORA3LMNACYP2C9CYP2C19CYP3A4
SCHEMBL8595275 0.87 HTT (0.53) ADORA3LMNACYP2C9CYP2C19CYP3A4
SCHEMBL8595272 0.87 HTT (0.53) ADORA3LMNACYP2C9CYP2C19CYP3A4
SCHEMBL8595500 0.86 LMNA (0.76) ADORA3LMNACYP2C9CYP2C19CYP3A4
SCHEMBL9872633 0.86 CYP3A4 (0.54) ADORA3LMNACYP2C9CYP2C19CYP3A4
SCHEMBL9872624 0.86 CYP3A4 (0.54) ADORA3LMNACYP2C9CYP2C19CYP3A4
SCHEMBL8595497 0.86 LMNA (0.76) ADORA3LMNACYP2C9CYP2C19CYP3A4
SCHEMBL10495738 0.86 LMNA (0.76) ADORA3LMNACYP2C9CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5011848-A Cardiovascular disorders, hypotensive agents GLAXO, S.P.A. (IT) 1991-04-30 US disclosed
US-4801599-A CARDIOVASCULAR DISORDERS, HYPOTENSIVE AGENTS GLAXO S.P.A. (IT) 1989-01-31 US disclosed