SCHEMBL9871600

SCHEMBL9871600

Cc1nc2c(Cl)nnc(O)c2n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 9/20 0.38
AGTR2 P50052 7/20 0.38
PDE10A Q9Y233 1/20 0.35
ABCC4 O15439 1/20 0.34
ABCB11 O95342 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9873895 0.93 AGTR1 (0.40) AGTR1AGTR2PDE10A
SCHEMBL9871897 0.92 AGTR1 (0.41) AGTR1AGTR2PDE10A
SCHEMBL9874151 0.90 AGTR1 (0.40) AGTR1AGTR2
SCHEMBL9873762 0.90 AGTR1 (0.38) AGTR1AGTR2PDE10A
SCHEMBL9872000 0.89 AGTR1 (0.39) AGTR1AGTR2
SCHEMBL9874580 0.89 AGTR2 (0.37) AGTR1AGTR2
SCHEMBL9871993 0.88 AGTR1 (0.38) AGTR1AGTR2
SCHEMBL9873634 0.88 AGTR1 (0.37) AGTR1AGTR2PDE10A
SCHEMBL9873077 0.88 AGTR1 (0.35) AGTR1AGTR2ABCC4ABCB11PDE3B
SCHEMBL9874478 0.88 AGTR1 (0.37) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019715-A1 1H-SUBSTITUTED-IMIDAZO[4,5-d]PYRIDAZINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1991-12-26 WO disclosed