SCHEMBL9871855

SCHEMBL9871855

C=CC(O)CC(=O)CC(=O)OCC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.48
MGAM O43451 1/20 0.48
SI P14410 1/20 0.48
MGAM2 Q2M2H8 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.37
ALDH1A1 P00352 3/20 0.36
TRPA1 O75762 1/20 0.36
CYP1A2 P05177 1/20 0.36
KMT2A Q03164 2/20 0.35
POLB P06746 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
NR1I2 O75469 1/20 0.33
PGR P06401 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
PTGS2 P35354 1/20 0.33
PDE4D Q08499 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6118705 0.85 GAA (0.44) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL9754935 0.83 TSHR (0.41) GAAMGAMSIMGAM2ALDH1A1
SCHEMBL31260805 0.77 GAA (0.56) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL9870922 0.75 CYP1A2 (0.40) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL14283521 0.75 CYP1A2 (0.40) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL15344 0.75 GAA (0.58) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL13530805 0.74
SCHEMBL9005312 0.74 GAA (0.52) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL959397 0.74 GAA (0.52) GAAMGAMSIMGAM2L3MBTL1
SCHEMBL155563 0.73 GAA (0.78) GAAMGAMSIMGAM2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997837-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-05 US disclosed
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed
EP-0306929-A2 6-[[(Substituted)pyridin-3-YL]alkyl]-and alkenyl]-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1989-03-15 EP disclosed
US-4650890-A Preparation of olefinic compounds and intermediates thereof SANDOZ CORP. (US) 1987-03-17 US disclosed