SCHEMBL9872202

SCHEMBL9872202

CCc1nc(CC)c(C(=O)O)c(-c2ccc(F)cc2)c1COC1CCCCO1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 2/20 0.42
DPP4 P27487 3/20 0.41
DPP8 Q6V1X1 2/20 0.41
DPP9 Q86TI2 2/20 0.41
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
CREBBP Q92793 2/20 0.35
FABP3 P05413 1/20 0.33
FABP4 P15090 1/20 0.33
FABP5 Q01469 1/20 0.33
DHODH Q02127 2/20 0.33
EP300 Q09472 1/20 0.33
ALDH1A1 P00352 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
GCGR P47871 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9879298 0.91 ADORA3 (0.41) ADORA3MEN1KMT2AL3MBTL1CREBBP
SCHEMBL9265733 0.76 GCGR (0.50) MEN1KMT2AL3MBTL1ALDH1A1GCGR
SCHEMBL8114161 0.75 KDM4E (0.36) MEN1KMT2ACREBBPEP300ALDH1A1
SCHEMBL9872670 0.75 ADORA3 (0.32) ADORA3MEN1KMT2AALDH1A1
SCHEMBL9872661 0.75 HMGCR (0.35) ADORA3MEN1KMT2ACREBBPALDH1A1
SCHEMBL9870568 0.74 DPP4 (0.50) DPP4DPP8DPP9FABP3FABP4
SCHEMBL27525559 0.74 PRKAA2 (0.51) DPP4DPP8DPP9FABP3FABP4
SCHEMBL6958480 0.72 GCGR (0.61) GCGR
SCHEMBL6949644 0.71 GCGR (0.41) GCGR
SCHEMBL2647574 0.71 PRKAA2 (0.47) DPP4DPP8DPP9FABP4FABP5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4997837-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1991-03-05 US disclosed
US-4906624-A 6-(((Substituted)pyridin-3-yl)alkyl)-and alkenyl)-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1990-03-06 US disclosed
EP-0306929-A2 6-[[(Substituted)pyridin-3-YL]alkyl]-and alkenyl]-tetrahydro-4-hydroxypyran-2-one inhibitors of cholesterol biosynthesis WARNER-LAMBERT COMPANY (US) 1989-03-15 EP disclosed