SCHEMBL9873313

SCHEMBL9873313

OC1Cc2ccccc2Sc2ccccc21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 11/20 0.41
HRH1 P35367 3/20 0.41
HTR2C P28335 3/20 0.41
TP53 P04637 3/20 0.41
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 3/20 0.41
DRD4 P21917 2/20 0.41
CYP2C19 P33261 2/20 0.41
NPC1 O15118 2/20 0.41
MTOR P42345 2/20 0.41
RAB9A P51151 2/20 0.41
NFKB1 P19838 2/20 0.41
THPO P40225 2/20 0.41
KCNK9 Q9NPC2 2/20 0.41
TSHR P16473 1/20 0.41
HIF1A Q16665 1/20 0.41
HTR7 P34969 3/20 0.40
MAPT P10636 3/20 0.40
SMN1; SMN2 Q16637 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11705882 0.82 HTR7 (0.40) DRD2HRH1HTR2CTP53CYP1A2
SCHEMBL11707106 0.82 HTR7 (0.40) DRD2HRH1HTR2CTP53CYP1A2
SCHEMBL8168724 0.82 HRH1 (0.50) DRD2HRH1HTR2CTP53CYP1A2
SCHEMBL11009156 0.82 HTR2C (0.36) DRD2HRH1HTR2CTP53CYP1A2
SCHEMBL11706143 0.82 DRD2 (0.41) DRD2HRH1HTR2CTP53CYP1A2
SCHEMBL8171297 0.82 DRD2 (0.44) DRD2HRH1HTR2CTP53CYP1A2
SCHEMBL11486519 0.80 DRD2 (0.36) DRD2HRH1HTR2CTP53CYP1A2
SCHEMBL11479312 0.80 DRD2 (0.42) DRD2HRH1HTR2CTP53CYP1A2
SCHEMBL11703879 0.78 CYBB (0.44) DRD2HRH1HTR2CTP53CYP1A2
SCHEMBL11013573 0.78 NPSR1 (0.40) DRD2HRH1HTR2CTP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5006664-A Reacting 10,11-dihydro-10-hydroxybenz b,f!thiepin with an aminoalkylthiol in presence of boron trifluoride etherate and solvent; antidepressant, analgesic, anticonvulsant HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-04-09 US claimed
US-5006664-A Reacting 10,11-dihydro-10-hydroxybenz b,f!thiepin with an aminoalkylthiol in presence of boron trifluoride etherate and solvent; antidepressant, analgesic, anticonvulsant HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1991-04-09 US disclosed
US-4775672-A ANTIDEPRESSANTS, ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1988-10-04 US disclosed
US-4775683-A ANTIDEPRESSANTS, ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1988-10-04 US disclosed
US-4775682-A ANALGESICS, ANTIPRESSANTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1988-10-04 US disclosed
US-4771069-A ANTIDEPRESSANTS, ANALGESICS, ANTICONVULSANTS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1988-09-13 US disclosed
US-4766143-A ANTIDEPRESSANTS, ANTICONVULSANTS, ANALGESICS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1988-08-23 US disclosed
US-4668695-A ANTIDEPRESSANTS, ANALGESICS ANTICONVULSANTS HOECHST ROUSSEL PHARMACEUTICALS INC. (US) 1987-05-26 US disclosed