SCHEMBL9873330

SCHEMBL9873330

CC1=C(C(=O)OCCC#N)C(c2ccccc2OC(F)(F)F)C([N+](=O)[O-])=C(C)N1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 6/20 0.53
CACNA1C Q13936 6/20 0.53
CYP1A2 P05177 5/20 0.53
MAPT P10636 5/20 0.53
CYP3A4 P08684 4/20 0.53
CYP2C9 P11712 4/20 0.53
CYP2C19 P33261 4/20 0.53
TSHR P16473 3/20 0.53
NFKB1 P19838 3/20 0.53
CYP2D6 P10635 2/20 0.53
KMT2A Q03164 2/20 0.53
MEN1 O00255 1/20 0.53
CACNA1F O60840 3/20 0.41
CACNA1D Q01668 3/20 0.41
CACNA1S Q13698 3/20 0.41
ABCC4 O15439 2/20 0.41
ABCB11 O95342 2/20 0.41
LMNA P02545 2/20 0.41
ADORA2A P29274 2/20 0.41
ADORA1 P30542 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9875222 0.88 CACNA1C (0.56) ADORA3CACNA1CCYP1A2MAPTCYP3A4
SCHEMBL10516018 0.88 MAPT (0.43) ADORA3CACNA1CCYP1A2MAPTCYP3A4
SCHEMBL9879777 0.88 NR1I2 (0.54) ADORA3CACNA1CCYP1A2MAPTCYP3A4
SCHEMBL11005379 0.87 CYP1A2 (0.71) ADORA3CACNA1CCYP1A2MAPTCYP3A4
SCHEMBL9876069 0.87 CACNA1C (0.55) ADORA3CACNA1CCYP1A2MAPTCYP3A4
SCHEMBL9876125 0.86 CACNA1C (0.54) ADORA3CACNA1CCYP1A2MAPTCYP3A4
SCHEMBL9875740 0.86 CACNA1C (0.54) ADORA3CACNA1CCYP1A2MAPTCYP3A4
SCHEMBL9875212 0.86 CACNA1C (0.54) ADORA3CACNA1CCYP1A2MAPTCYP3A4
SCHEMBL11009095 0.84 ADORA3 (0.74) ADORA3CACNA1CCYP1A2MAPTCYP3A4
SCHEMBL9879946 0.83 CACNA1C (0.50) ADORA3CACNA1CCYP1A2MAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008279-A Circulation-active fluoromethoxyphenyl dihydropyridine compounds BAYER AKTIENGESELLSCHAFT (DE) 1991-04-16 US disclosed