SCHEMBL9879946

SCHEMBL9879946

CC1=C(C(=O)OCCN2CCCCC2)C(c2ccccc2OC(F)(F)F)C([N+](=O)[O-])=C(C)N1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 9/20 0.50
ADORA3 P0DMS8 5/20 0.50
MAPT P10636 5/20 0.50
CYP1A2 P05177 4/20 0.50
CYP3A4 P08684 4/20 0.50
CYP2C9 P11712 4/20 0.50
CYP2C19 P33261 4/20 0.50
TSHR P16473 2/20 0.50
NFKB1 P19838 2/20 0.50
MEN1 O00255 2/20 0.50
CYP2D6 P10635 2/20 0.50
KMT2A Q03164 2/20 0.50
CACNA1F O60840 7/20 0.44
CACNA1D Q01668 7/20 0.44
CACNA1S Q13698 7/20 0.44
ADRA1A P35348 4/20 0.43
ADRA2A P08913 3/20 0.43
ADRA2B P18089 3/20 0.43
ADRA2C P18825 3/20 0.43
ADRA1D P25100 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10515418 0.89 CACNA1C (0.41) CACNA1CADORA3MAPTCYP1A2CYP3A4
SCHEMBL9875415 0.88 NR1I2 (0.51) CACNA1CADORA3MAPTCYP1A2CYP3A4
SCHEMBL9875222 0.85 CACNA1C (0.56) CACNA1CADORA3MAPTCYP1A2CYP3A4
SCHEMBL9876069 0.84 CACNA1C (0.55) CACNA1CADORA3MAPTCYP1A2CYP3A4
SCHEMBL9876125 0.83 CACNA1C (0.54) CACNA1CADORA3MAPTCYP1A2CYP3A4
SCHEMBL9873330 0.83 ADORA3 (0.53) CACNA1CADORA3MAPTCYP1A2CYP3A4
SCHEMBL9875740 0.83 CACNA1C (0.54) CACNA1CADORA3MAPTCYP1A2CYP3A4
SCHEMBL9875212 0.83 CACNA1C (0.54) CACNA1CADORA3MAPTCYP1A2CYP3A4
SCHEMBL11009095 0.81 ADORA3 (0.74) CACNA1CADORA3MAPTCYP1A2CYP3A4
SCHEMBL9875844 0.80 ADORA3 (0.50) CACNA1CADORA3MAPTCYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008279-A Circulation-active fluoromethoxyphenyl dihydropyridine compounds BAYER AKTIENGESELLSCHAFT (DE) 1991-04-16 US disclosed