SCHEMBL9874157

SCHEMBL9874157

Cc1nc2c(SCc3ccccc3)nnc(SCc3ccccc3)c2n1Cc1ccc(-c2ccccc2C(=O)O)cc1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AGTR1 P30556 10/20 0.52
AGTR2 P50052 10/20 0.52
PDE7A Q13946 1/20 0.51
PDE7B Q9NP56 1/20 0.51
PPARG P37231 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9871735 0.94 AGTR1 (0.49) AGTR1AGTR2PDE7APDE7BPPARG
SCHEMBL9872915 0.91 PPARG (0.53) PPARG
SCHEMBL9873865 0.88 PDE7A (0.55) AGTR1AGTR2PDE7APDE7BPPARG
SCHEMBL9873844 0.87 PPARG (0.52) PPARG
SCHEMBL9871833 0.86 AGTR1 (0.50) AGTR1AGTR2PPARG
SCHEMBL9872953 0.86 AGTR2 (0.63) AGTR1AGTR2
SCHEMBL9873399 0.85 PPARG (0.51) AGTR1AGTR2PPARG
SCHEMBL9871430 0.85 PPARG (0.51) PPARG
SCHEMBL9874400 0.85 PPARG (0.50) PPARG
SCHEMBL9873272 0.83 AGTR1 (0.53) AGTR1AGTR2PDE7APDE7BPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991019715-A1 1H-SUBSTITUTED-IMIDAZO[4,5-d]PYRIDAZINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1991-12-26 WO disclosed