SCHEMBL9874162

SCHEMBL9874162

Cc1cccc(C)c1NC(=O)Nc1nnn(Cc2ccccc2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
RIPK1 Q13546 1/20 0.47
RAB9A P51151 4/20 0.45
NPC1 O15118 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
GAA P10253 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.44
ALDH1A1 P00352 2/20 0.44
SCN4A P35499 2/20 0.44
LMNA P02545 2/20 0.43
USP2 O75604 1/20 0.43
TSHR P16473 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ALOX15 P16050 1/20 0.43
HDAC6 Q9UBN7 1/20 0.42
KCNJ6 P48051 1/20 0.42
KCNJ5 P48544 1/20 0.42
KCNJ3 P48549 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9873553 0.85 SMN1; SMN2 (0.47) CYP1A2CYP2C9CYP2C19RIPK1RAB9A
SCHEMBL9872284 0.80 RAB9A (0.46) CYP1A2CYP2C9CYP2C19RAB9ANPC1
SCHEMBL9872449 0.76 MAPK1 (0.45) CYP1A2CYP2C9CYP2C19RAB9ASMN1; SMN2
SCHEMBL26077550 0.70 RAB9A (0.54) CYP1A2CYP2C9CYP2C19RIPK1RAB9A
SCHEMBL30051979 0.70 MAPT (0.67) CYP1A2CYP2C9CYP2C19RAB9ASMN1; SMN2
SCHEMBL22589844 0.69 HDAC6 (0.60) CYP1A2CYP2C9CYP2C19RAB9ANPC1
SCHEMBL9133647 0.68 AURKA (0.57) RIPK1SMN1; SMN2ALDH1A1LMNA
SCHEMBL4405590 0.67 RAB9A (0.62) RAB9ANPC1SMN1; SMN2GAAL3MBTL1
SCHEMBL18366936 0.67 SMN1; SMN2 (0.52) CYP1A2RIPK1RAB9ANPC1SMN1; SMN2
SCHEMBL6277857 0.67 MEN1 (0.65) SMN1; SMN2GAAALDH1A1SCN4ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5073565-A Atherosclerosis, anticholesterol WARNER-LAMBERT COMPANY (US) 1991-12-17 US disclosed
WO-1991017150-A1 TETRAZOLE UREA AND THIOUREA ACAT INHIBITORS WARNER-LAMBERT COMPANY (US) 1991-11-14 WO disclosed