SCHEMBL9875466

SCHEMBL9875466

Nc1c2c(nc3cc(F)ccc13)CCCC2O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 3/20 0.67
CYP1A2 P05177 1/20 0.67
CYP2C9 P11712 1/20 0.67
TSHR P16473 1/20 0.67
ALDH1A1 P00352 1/20 0.67
NR3C1 P04150 1/20 0.67
KCNH2 Q12809 1/20 0.67
BCHE P06276 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10845949 0.90 ACHE (0.67) ACHECYP1A2CYP2C9TSHRALDH1A1
SCHEMBL9654428 0.84 ACHE (0.67) ACHECYP1A2CYP2C9TSHRALDH1A1
SCHEMBL9651915 0.84 ACHE (0.67) ACHECYP1A2CYP2C9TSHRALDH1A1
SCHEMBL9874918 0.84 CYP1A2 (0.63) ACHECYP1A2CYP2C9TSHRALDH1A1
SCHEMBL9875350 0.81 ACHE (0.63) ACHECYP1A2CYP2C9TSHRALDH1A1
Velnacrine SCHEMBL194467 0.81 CYP1A2 (1.00) ACHECYP1A2CYP2C9TSHRALDH1A1
SCHEMBL10286366 0.79 ACHE (0.67) ACHECYP1A2CYP2C9TSHRALDH1A1
SCHEMBL10846147 0.77 ACHE (0.69) ACHECYP1A2CYP2C9TSHRALDH1A1
SCHEMBL9685394 0.77 ACHE (0.69) ACHECYP1A2CYP2C9TSHRALDH1A1
SCHEMBL10351769 0.77 BCHE (0.48) ACHECYP1A2CYP2C9TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4695573-A COGNITION ACTIVATORS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-09-22 US claimed
EP-2681554-B1 BLOOD COLLECTION DEVICE CONTAINING LYSOPHOSPHOLIPASE INHIBITOR BECTON DICKINSON CO (US) 2017-08-09 EP disclosed
US-9459187-B2 Blood collection device containing lysophospholipase inhibitor BECTON, DICKINSON AND COMPANY (US) 2016-10-04 US disclosed
CN-104244902-A Sample collection devices with blood stabilizing agents BECTON DICKINSON CO 2014-12-24 CN disclosed
EP-2809289-A1 SAMPLE COLLECTION DEVICES WITH BLOOD STABILIZING AGENTS Becton, Dickinson and Company (US) 2014-12-10 EP disclosed
US-20140030754-A1 BLOOD COLLECTION DEVICE CONTAINING LYSOPHOSPHOLIPASE INHIBITOR BECTON, DICKINSON AND COMPANY (US) 2014-01-30 US disclosed
CN-203203992-U Blood collection device containing lysophospholipase inhibitor BECTON DICKINSON CO 2013-09-18 CN disclosed
US-20130209985-A1 SAMPLE COLLECTION DEVICES WITH BLOOD STABILIZING AGENTS BECTON, DICKINSON AND COMPANY 2013-08-15 US disclosed
WO-2013116702-A1 SAMPLE COLLECTION DEVICES WITH BLOOD STABILIZING AGENTS BECTON, DICKINSON AND COMPANY (US) 2013-08-08 WO disclosed
EP-0179383-B1 9-AMINO-1,2,3,4-TETRAHYDROACRIDIN-1-OL AND RELATED COMPOUNDS, A PROCESS FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1991-05-29 EP disclosed
US-4839364-A ALZHEIMER*S DISEASE; CHOLINESTERASE INHIBITORS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1989-06-13 US disclosed
US-4835275-A Method of preparing 9-amino-1,2,3,4,-tetrahydroacridin-1-ones and related compounds HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1989-05-30 US disclosed
US-4754050-A COGNITION ACTIVATORS HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1988-06-28 US disclosed
US-4695573-A COGNITION ACTIVATORS HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1987-09-22 US disclosed
EP-0179383-A2 9-Amino-1,2,3,4-tetrahydroacridin-1-ol and related compounds, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1986-04-30 EP disclosed