SCHEMBL9875972

SCHEMBL9875972

CCCCCC=CCc1ccc(C#N)cc1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.53
HSD17B10 Q99714 1/20 0.53
CYP2A6 P11509 1/20 0.48
LOXL2 Q9Y4K0 2/20 0.42
CYP19A1 P11511 3/20 0.41
KCNH2 Q12809 6/20 0.38
MGLL Q99685 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9875970 1.00 TSHR (0.53) TSHRHSD17B10CYP2A6LOXL2CYP19A1
SCHEMBL9827715 0.78 TSHR (0.46) TSHRHSD17B10CYP2A6KCNH2MGLL
SCHEMBL9827727 0.78 TSHR (0.46) TSHRHSD17B10CYP2A6KCNH2MGLL
SCHEMBL9827722 0.78 TSHR (0.46) TSHRHSD17B10CYP2A6KCNH2MGLL
SCHEMBL24916718 0.78 ALDH1A1 (0.45) TSHRHSD17B10CYP2A6MGLL
SCHEMBL18364694 0.78 ALDH1A1 (0.58) TSHRHSD17B10MGLL
SCHEMBL9401077 0.77 TRPV1 (0.40) KCNH2MGLL
SCHEMBL20421301 0.77 TOP1 (0.41) KCNH2
SCHEMBL9401079 0.77 TRPV1 (0.40) KCNH2MGLL
SCHEMBL20421302 0.77 TOP1 (0.41) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991015473-A1 LEUCOTRIENE ANTAGONISTS, A PREPARATION METHOD THEREFOR AND THERAPEUTIC USES THEREOF LABORATOIRES FOURNIER S.C.A. (FR) 1991-10-17 WO disclosed