SCHEMBL9877236

SCHEMBL9877236

CN(O)C(=O)c1ccc(NCc2ccccc2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.63
CA2 P00918 1/20 0.63
HDAC3 O15379 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC2 Q92769 1/20 0.55
NCOR2 Q9Y618 1/20 0.55
HTT P42858 2/20 0.53
FFAR1 O14842 2/20 0.53
FFAR4 Q5NUL3 1/20 0.53
HIF1A Q16665 1/20 0.51
ALDH1A1 P00352 5/20 0.50
CYP1A2 P05177 4/20 0.50
CYP2D6 P10635 4/20 0.50
USP2 O75604 2/20 0.48
CYP3A4 P08684 2/20 0.48
MAPK1 P28482 1/20 0.48
HPGD P15428 2/20 0.47
LMNA P02545 1/20 0.47
TSHR P16473 1/20 0.47
CYP2C19 P33261 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10411601 0.86 FFAR1 (0.50) CA1CA2FFAR1FFAR4HIF1A
SCHEMBL9877862 0.84 HDAC8 (0.53) FFAR1HIF1AMEN1KMT2A
SCHEMBL10412444 0.82 ALOX5 (0.49) HDAC1ALDH1A1CYP1A2CYP2D6CYP3A4
SCHEMBL5604560 0.80 CA1 (0.71) CA1CA2HDAC3HDAC1HDAC2
SCHEMBL1446643 0.80 CA1 (0.70) CA1CA2HDAC3HDAC1HDAC2
SCHEMBL2742815 0.80 CA1 (0.70) CA1CA2HDAC3HDAC1HDAC2
SCHEMBL11881329 0.78 CA1 (0.68) CA1CA2HDAC3HDAC1HDAC2
SCHEMBL18415526 0.78 CA1 (1.00) CA1CA2HDAC3HDAC1HDAC2
SCHEMBL9696433 0.78 CA1 (0.67) CA1CA2HDAC3HDAC1HDAC2
SCHEMBL10411587 0.77 TRPV1 (0.48) HDAC1FFAR1ALDH1A1NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5036157-A Hydroxamic acid derivatives, lipoxygenase and cyclooxygenase inhibitors, anticoagulants, antiinflammatory agents BURROUGHS WELLCOME CO. 1991-07-30 US disclosed
US-4977188-A Hydroamic acid derivatives BURROUGHS WELLCOME CO. (US) 1990-12-11 US disclosed
WO-1990001929-A1 NEW MEDICAL USE THE WELLCOME FOUNDATION LIMITED (GB) 1990-03-08 WO disclosed
US-4738986-A CYCLOOXYGENASE, LIDOXYGENASE INHIBITORS BURROUGHS WELLCOME CO. (US) 1988-04-19 US disclosed
EP-0196184-A2 Aryl derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1986-10-01 EP disclosed