SCHEMBL9878041

SCHEMBL9878041

O=C(c1ccc(C(F)(F)F)cc1)n1ccnc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.47
HPGD P15428 1/20 0.47
TSHR P16473 1/20 0.47
KMT2A Q03164 1/20 0.47
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
SLC6A7 Q99884 1/20 0.46
CD38 P28907 1/20 0.42
SRD5A2 P31213 1/20 0.42
NOS1 P29475 1/20 0.41
CYP19A1 P11511 1/20 0.41
GAA P10253 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HIF1A Q16665 1/20 0.41
EPAS1 Q99814 1/20 0.41
MCHR1 Q99705 1/20 0.41
GSK3B P49841 2/20 0.41
PTPN1 P18031 1/20 0.41
EPHX2 P34913 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13028401 0.88 ESR1 (0.38) MEN1HPGDTSHRKMT2ACES2
SCHEMBL9807751 0.86 CYP19A1 (0.46) CYP19A1TDP1
SCHEMBL13028410 0.84 CYP3A4 (0.41) MEN1HPGDKMT2ACYP19A1TDP1
SCHEMBL30580646 0.81 LTA4H (0.47) KMT2ACES2CES1SLC6A7CYP19A1
SCHEMBL13028408 0.81 ADH5 (0.51) TSHRSLC6A7CYP19A1
SCHEMBL31388182 0.80 CYP19A1 (0.52) MEN1KMT2ACYP19A1EPHX2
SCHEMBL18280916 0.80 ADH5 (0.54) MEN1TSHRKMT2ACYP19A1
SCHEMBL9879507 0.78 LSS (0.47) KMT2ACES2CES1SLC6A7CYP19A1
SCHEMBL4808545 0.78 CYP19A1 (0.48) HPGDCES2CES1CYP19A1GAA
SCHEMBL11106769 0.78 MAOB (0.46) KMT2ACES2CES1SLC6A7CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991012255-A1 THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1991-08-22 WO disclosed