SCHEMBL9878243

SCHEMBL9878243

COc1cc(OC)c2c(c1)C(=O)c1cc(C)cc(OC)c1C2=O

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.83
CYP1A2 P05177 2/20 0.83
CYP3A4 P08684 2/20 0.83
ELANE P08246 9/20 0.64
MAPT P10636 2/20 0.64
ALOX15 P16050 2/20 0.64
KDM4E B2RXH2 1/20 0.64
GLA P06280 1/20 0.64
HPGD P15428 1/20 0.64
ACLY P53396 2/20 0.46
ACHE P22303 1/20 0.44
EPHX2 P34913 3/20 0.43
PIM1 P11309 2/20 0.41
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
PTP4A3 O75365 1/20 0.41
GMNN O75496 1/20 0.41
LMNA P02545 1/20 0.41
ESR1 P03372 1/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16226679 0.91 ALDH1A1 (1.00) ALDH1A1CYP1A2CYP3A4ELANEMAPT
SCHEMBL16226368 0.89 ELANE (0.83) ALDH1A1CYP1A2CYP3A4ELANEMAPT
SCHEMBL16227337 0.89 ELANE (0.83) ALDH1A1CYP1A2CYP3A4ELANEMAPT
SCHEMBL16226349 0.81 ELANE (0.60) ALDH1A1CYP1A2CYP3A4ELANEMAPT
SCHEMBL16226869 0.81 ALDH1A1 (0.80) ALDH1A1CYP1A2CYP3A4ELANEMAPT
SCHEMBL27921217 0.81 ALDH1A1 (0.74) ALDH1A1CYP1A2CYP3A4ELANEMAPT
SCHEMBL9878296 0.80 ELANE (0.60) ALDH1A1CYP1A2CYP3A4ELANEMAPT
SCHEMBL27882221 0.80 ALDH1A1 (0.77) ALDH1A1CYP1A2CYP3A4ELANEMAPT
SCHEMBL6905135 0.79 ALDH1A1 (0.77) ALDH1A1CYP1A2CYP3A4ELANEMAPT
SCHEMBL16227270 0.79 ALDH1A1 (0.70) ALDH1A1CYP1A2CYP3A4ELANEMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115850257-A Synthetic method of emodin amide derivatives containing coumarin thiazole and application of emodin amide derivatives in resisting marine vibrio 江苏海洋大学 2023-03-28 CN claimed
CN-112480031-B Emodin amide derivatives containing 1,3, 4-thiadiazole, and synthesis method and application thereof 江苏海洋大学 2022-05-20 CN claimed
CN-112480031-A Emodin amide derivatives containing 1,3, 4-thiadiazole, and synthesis method and application thereof 江苏海洋大学 2021-03-12 CN claimed
CN-102241598-B Monohydroxy emodin dioctyl quaternary ammonium salt with anticancer activity UNIV FUZHOU 2014-07-09 CN claimed
CN-103819350-A Chemical modification method capable of improving producing ability of reactive oxygen species (ROS) of rheum emodin UNIV FUZHOU 2014-05-28 CN claimed
CN-101941914-B Hydroxyl whole-protection didecyl quaternary ammonium with anti-tumor activity and preparation method thereof UNIV FUZHOU 2013-08-07 CN claimed
CN-101967105-B Beta-hydroxy protected didecyl quaternary ammonium salt with anticancer activity and preparation method thereof UNIV FUZHOU 2013-04-17 CN claimed
CN-102363044-B Application of three anthraquinone substances of targeted mitochondria as nasopharyngeal darcinoma radiosensitizers HOU HUAXIN 2013-03-20 CN claimed
CN-102649765-A Emodin di-n-octyl quaternary ammonium salt with anti-leukemia activity and preparation method thereof FUJIAN MEDICAL UNIVERSITY UNION HOSPITAL 2012-08-29 CN claimed
CN-102614158-A Emodin derivative with antitumor activity and preparation method thereof UNIV FUZHOU 2012-08-01 CN claimed
CN-102363044-A Application of three anthraquinone substances of targeted mitochondria as nasopharyngeal darcinoma radiosensitizers HUAXIN HOU 2012-02-29 CN claimed
CN-102249941-A Monohydroxy di(n-decyl) emodin quaternary ammonium salt with anticancer activity UNIV FUZHOU 2011-11-23 CN claimed
CN-102241598-A Monohydroxy emodin dioctyl quaternary ammonium salt with anticancer activity UNIV FUZHOU 2011-11-16 CN claimed
CN-102173997-A Liver cancer, gastric cancer and cervical cancer-resistant archen derivative and preparation method thereof UNIV FUZHOU 2011-09-07 CN claimed
CN-101967105-A Beta-hydroxy protected didecyl quaternary ammonium salt with anticancer activity and preparation method thereof UNIV FUZHOU 2011-02-09 CN claimed
CN-101941914-A Hydroxyl whole-protection didecyl quaternary ammonium with anti-tumor activity and preparation method thereof UNIV FUZHOU 2011-01-12 CN claimed
CN-115850257-A Synthetic method of emodin amide derivatives containing coumarin thiazole and application of emodin amide derivatives in resisting marine vibrio 江苏海洋大学 2023-03-28 CN disclosed
CN-112480031-B Emodin amide derivatives containing 1,3, 4-thiadiazole, and synthesis method and application thereof 江苏海洋大学 2022-05-20 CN disclosed
US-5053431-A Antitumor-anticarcinogenic agents SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1991-10-01 US disclosed
WO-1990008759-A1 DERIVATIVES OF CHRYSOPHANOL SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 1990-08-09 WO disclosed