SCHEMBL9878449

SCHEMBL9878449

Cc1ccccc1Nc1nc2c(c(=O)[nH]1)CCCC2

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.66
SMN1; SMN2 Q16637 3/20 0.66
NPC1 O15118 2/20 0.66
RAB9A P51151 2/20 0.66
ALPL P05186 1/20 0.59
ALPI P09923 1/20 0.59
ALPG P10696 1/20 0.59
TP53 P04637 1/20 0.58
OPRK1 P41145 1/20 0.58
HPGD P15428 4/20 0.57
PDE9A O76083 2/20 0.56
PKM P14618 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
CXCR2 P25025 2/20 0.52
KDM4E B2RXH2 1/20 0.50
ALDH1A1 P00352 1/20 0.50
TSHR P16473 1/20 0.50
HSD17B10 Q99714 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9878603 0.91 SMN1; SMN2 (0.56) MAPTSMN1; SMN2NPC1RAB9AALPL
SCHEMBL9878904 0.82 MAPT (0.75) MAPTSMN1; SMN2NPC1RAB9AALPL
SCHEMBL9878731 0.82 MEN1 (0.51) MAPTSMN1; SMN2NPC1RAB9AALPL
SCHEMBL9878442 0.78 MEN1 (0.53) MAPTSMN1; SMN2NPC1RAB9ATP53
SCHEMBL9878899 0.78 MEN1 (0.53) MAPTSMN1; SMN2NPC1RAB9AALPL
SCHEMBL9879015 0.76 KMT2A (0.60) MAPTSMN1; SMN2NPC1RAB9AHPGD
SCHEMBL9776663 0.73 KMT2A (0.65) MAPTSMN1; SMN2NPC1RAB9AHPGD
SCHEMBL31087175 0.73 HPGD (1.00) HPGDPKML3MBTL1
SCHEMBL16981701 0.72 PDE9A (1.00) PDE9A
SCHEMBL9878600 0.71 MEN1 (0.45) MAPTSMN1; SMN2NPC1RAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991018887-A1 DIAMINOPYRIMIDINE COMPOUNDS SMITHKLINE BEECHAM INTERCREDIT B.V. (NL) 1991-12-12 WO disclosed