SCHEMBL9879148

SCHEMBL9879148

C=CCOC(=O)C(CCC)c1ccccc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
HSD17B10 Q99714 4/20 0.50
TSHR P16473 2/20 0.50
CYP3A4 P08684 1/20 0.42
POLB P06746 3/20 0.35
KDM4E B2RXH2 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
PKM P14618 1/20 0.35
GAA P10253 2/20 0.33
RHOA P61586 1/20 0.33
MAPT P10636 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
GABRP O00591 1/20 0.33
GABRD O14764 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB1 P18505 1/20 0.33
GABRG2 P18507 1/20 0.33
GABRB3 P28472 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9879547 0.85 CYP3A4 (0.43) ALDH1A1HSD17B10TSHRCYP3A4POLB
SCHEMBL28235232 0.80 CYP2C19 (0.49) ALDH1A1HSD17B10TSHRCYP3A4KDM4E
SCHEMBL9879417 0.80 ALDH1A1 (0.48) ALDH1A1TSHRCYP3A4POLBKDM4E
SCHEMBL28755969 0.77 THRB (0.41) ALDH1A1HSD17B10TSHRCYP3A4GAA
SCHEMBL19951679 0.76 PPARG (0.39) ALDH1A1HSD17B10TSHRCYP3A4POLB
SCHEMBL9657053 0.76 ALDH1A1 (0.38) ALDH1A1HSD17B10CYP3A4POLBKDM4E
SCHEMBL27736942 0.76 EPHX1 (0.39) ALDH1A1HSD17B10CYP3A4POLBKDM4E
SCHEMBL1162115 0.76 PPARG (0.39) ALDH1A1HSD17B10TSHRCYP3A4POLB
SCHEMBL28755966 0.75 CYP3A4 (0.34) ALDH1A1HSD17B10TSHRCYP3A4KDM4E
Methane SCHEMBL28344019 0.75 PPARG (0.38) ALDH1A1HSD17B10TSHRCYP3A4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5008285-A Antiarthritic agent with low gastric irritability side effect HOECHST-ROUSSEL PHARMACEUTICALS, INC. (US) 1991-04-16 US disclosed
EP-0159684-B1 (6,11-DIHYDRO-11-OXODIBENZ(B,E)OXEPINYL)PENTANOIC ACIDS AND DERIVATIVES, A PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1989-09-27 EP disclosed
EP-0159684-A2 (6,11-Dihydro-11-oxodibenz(b,e)oxepinyl)pentanoic acids and derivatives, a process and intermediates for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1985-10-30 EP disclosed