SCHEMBL9891773

SCHEMBL9891773

Cc1cc(N2C(=O)CCC2C(C)C)ccc1F

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.36
HDAC8 Q9BY41 2/20 0.36
HDAC6 Q9UBN7 2/20 0.36
IDH1 O75874 4/20 0.35
MMP2 P08253 1/20 0.34
ADAMTS5 Q9UNA0 1/20 0.34
CCR1 P32246 1/20 0.33
CCR2 P41597 1/20 0.33
MDM2 Q00987 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4D Q08499 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
GFER P55789 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9891763 0.89 CCR1 (0.43) HDAC1HDAC8HDAC6CCR1CCR2
SCHEMBL9891772 0.89 BPTF (0.39) HDAC1HDAC8HDAC6CCR1CCR2
SCHEMBL9891760 0.85 KMT2A (0.45) CYP1A2CYP2C19
SCHEMBL9891767 0.83 CCR1 (0.43) CCR1CCR2MDM2
SCHEMBL9891766 0.82 IDO1 (0.38) HDAC1HDAC8HDAC6IDH1CYP1A2
SCHEMBL9893055 0.81 PARP1 (0.43) HDAC1HDAC8HDAC6MMP2ADAMTS5
SCHEMBL24415451 0.81 CREBBP (0.38) HDAC1HDAC8HDAC6CCR1CCR2
SCHEMBL9891770 0.81 PKM (0.46) GFER
SCHEMBL9891768 0.80 HTR7 (0.40)
SCHEMBL9891774 0.80 HDAC6 (0.32) HDAC1HDAC8HDAC6IDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8629157-B2 Pyrrolidine compounds which modulate the CB2 receptor BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-01-14 US disclosed
US-20120142677-A1 Pyrrolidine Compounds Which Modulate The CB2 Receptor BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120142677-A1 Pyrrolidine Compounds Which Modulate The CB2 Receptor CNR2, CNR1, OPRL1 HDAC1 1767/4885HDAC8 2405/4885HDAC6 1750/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.