SCHEMBL989255

SCHEMBL989255

CN1CCN=C1CCCCCCCCCCCCC1=NCCN1C

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
HTR1D P28221 1/20 0.42
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
NOS1 P29475 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2417762 0.98 ADRA2A (0.41) ADRA2AADRA2BADRA2CHTR1DCYP1A2
SCHEMBL10948416 0.92 ADRA2A (0.38) ADRA2AADRA2BADRA2CHTR1D
SCHEMBL6292172 0.92 ADRA2A (0.38) ADRA2AADRA2BADRA2CHTR1D
SCHEMBL2516256 0.92 ADRA2A (0.38) ADRA2AADRA2BADRA2CHTR1D
SCHEMBL6660516 0.87 HTR1D (0.40) ADRA2AADRA2BADRA2CHTR1D
SCHEMBL9398117 0.83 FAAH (0.42)
SCHEMBL9398124 0.83 FAAH (0.42)
SCHEMBL20052856 0.82
SCHEMBL7267539 0.80
SCHEMBL10619672 0.78 MIF (0.33) ADRA2AADRA2BADRA2CHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2275100-A2 Compounds with anti-parasitic activity and drugs containing said compounds Centre National de la Recherche Scientifique (CNRS) (FR) 2011-01-19 EP disclosed
EP-2266555-A2 Compounds with antiparasitic activity and medicines containing same Centre National de la Recherche Scientifique (CNRS) (FR) 2010-12-29 EP disclosed
EP-2260840-A2 Compounds with antiparasitic activity and medicines containing same Centre National de la Recherche Scientifique (CNRS) (FR) 2010-12-15 EP disclosed
EP-2260841-A2 Compounds with antiparasitic activity and medicines containing same Centre National de la Recherche Scientifique (CNRS) (FR) 2010-12-15 EP disclosed
EP-1524972-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY AND MEDICINES CONTAINING SAME CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2005-04-27 EP disclosed
WO-2004009068-A2 COMPOUNDS WITH ANTIPARASITIC ACTIVITY AND MEDICINES CONTAINING SAME CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2004-01-29 WO disclosed