SCHEMBL989952

SCHEMBL989952

C=C(CBr)c1ccc(F)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.48
CES1 P23141 2/20 0.48
MAOA P21397 5/20 0.43
MAOB P27338 5/20 0.43
PTPN1 P18031 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CHRNA1 P02708 1/20 0.34
CHRNG P07510 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
SLC6A2 P23975 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNA4 P43681 1/20 0.34
SLC6A3 Q01959 1/20 0.34
CHRND Q07001 1/20 0.34
PLA2G7 Q13093 1/20 0.33
KCNQ3 O43525 2/20 0.33
KCNQ2 O43526 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31368922 0.82 KCNQ3 (0.39) CES2CES1MAOAMAOBPTPN1
SCHEMBL16795682 0.81 CES2 (0.50) CES2CES1MAOAMAOBMEN1
SCHEMBL16795584 0.78 CES2 (0.44) CES2CES1PTPN1
SCHEMBL991185 0.78 HTT (0.56) MEN1KMT2AKCNQ3KCNQ2RAB9A
SCHEMBL2175225 0.76 PTPN1 (0.56) CES2CES1MAOAMAOBPTPN1
SCHEMBL16953016 0.75 CES2 (0.48) CES2CES1MAOAMAOBPTPN1
SCHEMBL29628387 0.75 PTPN1 (0.61) CES2CES1PTPN1MEN1KMT2A
SCHEMBL366866 0.75 PTPN1 (0.61) CES2CES1PTPN1MEN1KMT2A
SCHEMBL991358 0.71 GSK3B (0.56) CES2CES1MAOAMAOBGSK3B
SCHEMBL20938010 0.71 CES2 (0.54) CES2CES1MAOAMAOBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2480080-A1 PYRIDO[3,4-B]INDOLES AND METHODS OF USE Medivation Technologies, Inc. (US) 2012-08-01 EP disclosed
WO-2011038163-A1 PYRIDO[3,4-B]INDOLES AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2011-03-31 WO disclosed
EP-2274307-A1 BRIDGED HETEROCYCLIC COMPOUNDS AND METHODS OF USE Medivation Technologies, Inc. (US) 2011-01-19 EP disclosed
WO-2009120720-A1 BRIDGED HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES,INC. (US) 2009-10-01 WO disclosed
US-6025310-A RETAINING STABILITY FREE OF HYDROLYSIS FOR PROLONGED PERIOD OF TIME, COMPATIBLE WITH ORGANIC LUBRICANTS HAVING BENZENE RING AND PHOSPHAZINE RING KUBOTA CORPORATION (JP) 2000-02-15 US disclosed