Bicarbonate

Bicarbonate

SCHEMBL9899636

CC(C(C(=O)Nc1cc(CC2CC2)ccc1Cl)c1ccc(CC(F)(F)F)cc1)C(F)(F)F.O=C(O)O

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.41
SMN1; SMN2 Q16637 2/20 0.37
PDE2A O00408 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
PANK3 Q9H999 1/20 0.35
HDAC1 Q13547 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
MEN1 O00255 3/20 0.34
KDM4E B2RXH2 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
GAA P10253 2/20 0.34
HTT P42858 1/20 0.34
ALDH1A1 P00352 2/20 0.34
FAAH O00519 1/20 0.34
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
CTDSP1 Q9GZU7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL16735616 0.93 KMT2A (0.41) KMT2ASMN1; SMN2L3MBTL1PANK3TRPV1
Bicarbonate SCHEMBL16735635 0.91 KMT2A (0.47) KMT2ASMN1; SMN2L3MBTL1MEN1KDM4E
Bicarbonate SCHEMBL16735568 0.90 KMT2A (0.39) KMT2ASMN1; SMN2L3MBTL1PANK3TRPV1
Bicarbonate SCHEMBL16735651 0.89 KMT2A (0.41) KMT2ASMN1; SMN2PDE2AL3MBTL1PANK3
Bicarbonate SCHEMBL16735653 0.88 KMT2A (0.41) KMT2AL3MBTL1MEN1KDM4EGAA
SCHEMBL1931935 0.85 KMT2A (0.39) KMT2ASMN1; SMN2L3MBTL1HDAC1TRPV1
Bicarbonate SCHEMBL16735627 0.85 FFAR2 (0.38) UBE2MDCUN1D1CCR3
SCHEMBL1905649 0.85 SMN1; SMN2 (0.37) KMT2ASMN1; SMN2PDE2AL3MBTL1HDAC1
SCHEMBL1932256 0.85 KMT2A (0.39) KMT2ASMN1; SMN2L3MBTL1HDAC1TRPV1
SCHEMBL1932582 0.85 KMT2A (0.39) KMT2ASMN1; SMN2L3MBTL1HDAC1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649045-B1 SUBSTITUTED 1-BENZYLCYCLOALKYLCARBOXLIC ACIDS AND USE THEREOF BAYER IP GMBH (DE) 2015-05-27 EP disclosed
EP-2649045-A2 SUBSTITUTED 1-BENZYLCYCLOALKYLCARBOXLIC ACIDS AND USE THEREOF Bayer Intellectual Property GmbH (DE) 2013-10-16 EP disclosed
WO-2012076466-A2 SUBSTITUTED 1-BENZYLCYCLOALKYLCARBOXLIC ACIDS AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-06-14 WO disclosed