SCHEMBL9899768

SCHEMBL9899768

O=C(O)Nc1cnccc1-c1ccc(O)cc1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RPS6KA3 P51812 2/20 0.56
SLC22A12 Q96S37 1/20 0.46
GSK3B P49841 13/20 0.45
GSK3A P49840 12/20 0.45
JAK2 O60674 1/20 0.43
PIM1 P11309 1/20 0.43
CDK2 P24941 1/20 0.43
TYK2 P29597 1/20 0.43
SYK P43405 1/20 0.43
CDK5 Q00535 1/20 0.43
PRKCQ Q04759 1/20 0.43
AURKB Q96GD4 1/20 0.43
MAPT P10636 4/20 0.43
ALDH1A1 P00352 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9900438 0.87 RPS6KA3 (0.56) RPS6KA3SLC22A12ALDH1A1ALOX15TSHR
SCHEMBL16628650 0.76 GPBAR1 (0.47) GSK3BGSK3ATYK2TSHR
SCHEMBL5106705 0.76 ALDH1A1 (0.55) MAPTALDH1A1TSHR
SCHEMBL9915925 0.76 LPAR1 (0.52) RPS6KA3SLC22A12GSK3BGSK3AMAPT
SCHEMBL27426524 0.75 GSK3B (0.55) GSK3BGSK3AMAPTALDH1A1ALOX15
SCHEMBL12496930 0.75 GSK3A (0.55) GSK3BGSK3AALDH1A1ALOX15TSHR
SCHEMBL16702338 0.72 ATR (0.52) GSK3BGSK3AMAPT
SCHEMBL5826769 0.72 KDM4C (0.44) GSK3BGSK3AMAPT
SCHEMBL8946928 0.72 TAAR1 (0.60) GSK3BGSK3AMAPTTSHR
SCHEMBL15770896 0.72 PIK3C3 (0.44) GSK3BGSK3AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2648714-A2 LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AND USES THEREOF Amira Pharmaceuticals, Inc. (US) 2013-10-16 EP disclosed
WO-2012078593-A2 LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AND USES THEREOF AMIRA PHARMACEUTICALS, INC. (US) 2012-06-14 WO disclosed