SCHEMBL9899952

SCHEMBL9899952

CC(C(=O)O)(c1ccc(Cl)c(Cl)c1)C1CCCC1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 1/20 0.42
KEAP1 Q14145 1/20 0.41
NFE2L2 Q16236 1/20 0.41
SLC6A3 Q01959 2/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R2 Q8TE23 1/20 0.39
CHRM3 P20309 6/20 0.39
TSHR P16473 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
AR P10275 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
SSTR3 P32745 1/20 0.37
CHRM2 P08172 1/20 0.36
CHRM4 P08173 1/20 0.36
CHRM1 P11229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3554824 0.83 CHRM3 (0.44) KEAP1NFE2L2CHRM3MAPTCYP3A4
SCHEMBL2646811 0.80 SLC6A3 (0.41) SSTR4SLC6A3TAS1R3TAS1R2LMNA
SCHEMBL27770442 0.78 CHRM3 (0.45) KEAP1NFE2L2SLC6A3CHRM3TSHR
SCHEMBL4213705 0.77 KEAP1 (0.61) KEAP1NFE2L2CHRM3CYP2C9CHRM2
SCHEMBL4203042 0.77 KEAP1 (0.61) KEAP1NFE2L2CHRM3CYP2C9CHRM2
SCHEMBL4203592 0.77 KEAP1 (0.61) KEAP1NFE2L2CHRM3CYP2C9CHRM2
SCHEMBL9899047 0.76 CHRM3 (0.44) KEAP1NFE2L2CHRM3CYP3A4CYP2C9
SCHEMBL4247916 0.76 KEAP1 (0.47) KEAP1NFE2L2CHRM3CHRM2CHRM4
SCHEMBL7550366 0.76 MEN1 (0.44) CHRM3TSHRMAPTCYP3A4CYP2C9
SCHEMBL2788610 0.76 KEAP1 (0.59) KEAP1NFE2L2CHRM3CHRM2CHRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649045-B1 SUBSTITUTED 1-BENZYLCYCLOALKYLCARBOXLIC ACIDS AND USE THEREOF BAYER IP GMBH (DE) 2015-05-27 EP disclosed
EP-2649045-A2 SUBSTITUTED 1-BENZYLCYCLOALKYLCARBOXLIC ACIDS AND USE THEREOF Bayer Intellectual Property GmbH (DE) 2013-10-16 EP disclosed
WO-2012076466-A2 SUBSTITUTED 1-BENZYLCYCLOALKYLCARBOXLIC ACIDS AND USE THEREOF BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-06-14 WO disclosed