SCHEMBL9900075

SCHEMBL9900075

Cc1cccc(-c2nc(C(N)=O)co2)c1

nearest known ligand 0.68

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.68
HDAC1 Q13547 5/20 0.50
HDAC8 Q9BY41 5/20 0.50
HDAC6 Q9UBN7 5/20 0.50
PDE4B Q07343 9/20 0.48
SLC9A1 P19634 1/20 0.44
PARP1 P09874 1/20 0.44
DHODH Q02127 1/20 0.43
ENPP3 O14638 1/20 0.43
NPC1 O15118 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10029551 0.87 HDAC1 (0.51) ALDH1A1HDAC1HDAC8HDAC6PDE4B
SCHEMBL12377852 0.83 HDAC1 (0.51) ALDH1A1HDAC1HDAC8HDAC6PDE4B
SCHEMBL12377858 0.83 HSD17B1 (0.48) ALDH1A1HDAC1HDAC8HDAC6PDE4B
SCHEMBL12377859 0.83 HDAC1 (0.58) ALDH1A1HDAC1HDAC8HDAC6PDE4B
SCHEMBL28033118 0.81 ALDH1A1 (0.71) ALDH1A1HDAC1HDAC8HDAC6PDE4B
SCHEMBL893099 0.81 ALDH1A1 (1.00) ALDH1A1HDAC1HDAC8HDAC6PDE4B
SCHEMBL12377853 0.80 HDAC1 (0.54) ALDH1A1HDAC1HDAC8HDAC6PDE4B
SCHEMBL29502534 0.78 IRAK4 (0.62) ALDH1A1
SCHEMBL16896536 0.78 IRAK4 (0.62) ALDH1A1
Hydrochloric Acid SCHEMBL16896632 0.77 IRAK4 (0.62) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103380130-B Novel pyrazole and imidazole derivatives useful as orexin antagonists ACTELION PHARMACEUTICALS LTD 2015-06-17 CN disclosed
EP-2649068-A1 OXAZOLYL-METHYLETHER DERIVATIVES AS ALX RECEPTOR AGONISTS Actelion Pharmaceuticals Ltd. (CH) 2013-10-16 EP disclosed
WO-2012077049-A1 OXAZOLYL-METHYLETHER DERIVATIVES AS ALX RECEPTOR AGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2012-06-14 WO disclosed