SCHEMBL9900927

SCHEMBL9900927

CCOC(=O)C=C(ON(NC(=O)OCc1ccccc1)C(=N)C1CCC(F)(CO)CC1)C(=O)OCC

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.37
MAOB P27338 1/20 0.37
ALDH1A1 P00352 2/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 2/20 0.34
RORC P51449 1/20 0.34
CPB1 P15086 2/20 0.33
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
DPP4 P27487 1/20 0.32
KCNH2 Q12809 1/20 0.32
DPP7 Q9UHL4 1/20 0.32
LMNA P02545 1/20 0.32
LGMN Q99538 1/20 0.32
CTSL P07711 1/20 0.31
CYP3A4 P08684 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9942885 0.76 CTSS (0.38) KDM1AMAOBRORCCPB1SMN1; SMN2
SCHEMBL51559 0.69 CTSS (0.38) ALDH1A1GAATSHRRORCCPB1
SCHEMBL13924823 0.68 NR1H4 (0.49) ALDH1A1LMNA
SCHEMBL13657353 0.68 RORC (0.38) TSHRRORCCPB1SMN1; SMN2CTSL
SCHEMBL5528333 0.68 TLR2 (0.41) RORCLGMNCTSL
SCHEMBL63524 0.67 CTSS (0.37) ALDH1A1GAATSHRRORCCPB1
SCHEMBL13691697 0.67 CTSS (0.37) ALDH1A1GAATSHRRORCCPB1
SCHEMBL13657354 0.67 RORC (0.37) TSHRRORCCPB1SMN1; SMN2CTSL
SCHEMBL62654 0.66 CTSS (0.35) TSHRRORCCPB1CTSL
SCHEMBL13691437 0.66 CTSS (0.35) TSHRRORCCPB1CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2649077-A1 HIV INTEGRASE INHIBITORS Bristol-Myers Squibb Company (US) 2013-10-16 EP disclosed
WO-2012078834-A1 HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-06-14 WO disclosed