SCHEMBL9901327

SCHEMBL9901327

COc1cccc(COc2c(C)c(C)n(-c3ccnc(-c4ccnc(C(C)(C)O)n4)c3)c(=O)c2C)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.37
PKM P14618 1/20 0.37
MAOA P21397 1/20 0.37
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
MAPKAPK2 P49137 2/20 0.36
MAPKAPK5 Q8IW41 1/20 0.36
PIK3CA P42336 1/20 0.36
ROCK2 O75116 3/20 0.35
F10 P00742 1/20 0.35
PTGER1 P34995 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
ACHE P22303 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9901213 0.93 MAOB (0.38) MAOBPKMMAOAMTNR1AMTNR1B
SCHEMBL9902078 0.91 MAPKAPK2 (0.38) MAOBMAOAMAPKAPK2MAPKAPK5PIK3CA
SCHEMBL9109270 0.87 MAPKAPK2 (0.44) MAOBPKMMAOAMTNR1AMTNR1B
SCHEMBL9902659 0.87 MAPKAPK2 (0.38) MAOBPKMMAOAMTNR1AMTNR1B
SCHEMBL9902453 0.85 MAOB (0.36) MAOBPKMMAOAMTNR1AMTNR1B
SCHEMBL9905107 0.84 MAPKAPK2 (0.38) MAPKAPK2MAPKAPK5
SCHEMBL9110577 0.83 MAPKAPK5 (0.52) MAOBPKMMAOAMAPKAPK2MAPKAPK5
SCHEMBL9108095 0.82 MAPK14 (0.45) MAPKAPK2MAPKAPK5PIK3CAPTGER1SMN1; SMN2
SCHEMBL9905046 0.81 MAPKAPK2 (0.36) MAPKAPK2MAPKAPK5
SCHEMBL9111055 0.80 MAPKAPK2 (0.42) MAOBPKMMAOAMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2648516-A1 SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS Confluence Life Sciences, Inc. (US) 2013-10-16 EP disclosed
WO-2012078684-A1 SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS CONFLUENCE LIFE SCIENCES, INC. (US) 2012-06-14 WO disclosed