SCHEMBL9905002

SCHEMBL9905002

Nc1ccc(N2CCCCC2(I)C(=O)O)cc1C(F)(F)F

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 1/20 0.36
AR P10275 6/20 0.34
NOTUM Q6P988 6/20 0.33
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
FAAH O00519 1/20 0.32
FFAR4 Q5NUL3 1/20 0.31
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31
FFAR1 O14842 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
AOC3 Q16853 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2979456 0.81 CNR1 (0.42) IP6K1ARNOTUMNR1H2NR1H3
SCHEMBL13244521 0.73 CNR1 (0.42) ARNOTUMNR1H2NR1H3FFAR4
SCHEMBL3711951 0.71 HSD11B1 (0.44) NOTUMSMN1; SMN2
SCHEMBL962246 0.70 HTT (0.56) IP6K1ARNOTUMSMN1; SMN2NPSR1
SCHEMBL2012912 0.69 HTT (0.59) IP6K1ARNOTUMSMN1; SMN2NPSR1
SCHEMBL2052714 0.68 HSD11B1 (0.42) IP6K1ARNOTUMCNR1CNR2
SCHEMBL2053813 0.67 GAA (0.51) IP6K1ARNOTUMSMN1; SMN2NPSR1
SCHEMBL2969960 0.67 S100B (0.39) IP6K1ARNOTUM
SCHEMBL2978178 0.67 HSD11B1 (0.45) ARNOTUMCNR1CNR2
SCHEMBL2979182 0.66 AR (0.40) IP6K1ARNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072241-A9 4-OXO-1H-QUINOLINE-3-CARBOXAMIDES AS MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-06-14 WO disclosed