SCHEMBL9905385

SCHEMBL9905385

Cc1cc(C#Cc2cnc3cccnc3c2)cnc1N

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 2/20 0.43
NOS1 P29475 2/20 0.43
NOS2 P35228 2/20 0.43
PRMT5 O14744 1/20 0.39
MAP4K4 O95819 1/20 0.38
GRM5 P41594 2/20 0.35
ATAD2 Q6PL18 1/20 0.35
PDGFRB P09619 1/20 0.34
PDGFRA P16234 1/20 0.34
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
ALDH1A1 P00352 1/20 0.33
TGFBR1 P36897 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9902856 0.80 GRM5 (0.47) GRM5ATAD2PDGFRBPDGFRAALDH1A1
SCHEMBL9903498 0.80 GRM5 (0.46) GRM5PDGFRBPDGFRATGFBR1
SCHEMBL9903708 0.79 ABL1 (0.40) GRM5PDGFRBPDGFRAALDH1A1
SCHEMBL9903391 0.79 MTOR (0.45) PIK3CAMTOR
SCHEMBL23283107 0.78 GRM5 (0.49) NOS3NOS1NOS2MAP4K4GRM5
SCHEMBL9902619 0.78 GRM5 (0.51) GRM5PDGFRBPDGFRAALDH1A1
SCHEMBL9903420 0.78 GRM5 (0.55) GRM5PDGFRBPDGFRAALDH1A1
SCHEMBL9902735 0.76 PIK3CA (0.42) GRM5PDGFRBPDGFRAPIK3CAMTOR
SCHEMBL9902843 0.75 AAK1 (0.50) GRM5PIK3CAMTOR
SCHEMBL9903388 0.75 ALDH1A1 (0.39) GRM5PDGFRBALDH1A1TGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2462142-A1 METABOTROPIC GLUTAMATE RECEPTOR MODULATORS Merz Pharma GmbH & Co. KGaA (DE) 2012-06-13 EP claimed