SCHEMBL9908245

SCHEMBL9908245

CC(C)c1cc(C(C)(C)C)nn1CC(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.39
GRN P28799 4/20 0.36
SORT1 Q99523 4/20 0.36
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.33
FPR1 P21462 1/20 0.32
NPC1 O15118 1/20 0.32
PSEN1 P49768 2/20 0.31
PSEN2 P49810 2/20 0.31
APH1B Q8WW43 2/20 0.31
NCSTN Q92542 2/20 0.31
APH1A Q96BI3 2/20 0.31
PSENEN Q9NZ42 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
CNR1 P21554 2/20 0.31
CNR2 P34972 2/20 0.31
NPSR1 Q6W5P4 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9906363 0.81 GRN (0.39) GRNSORT1ALDH1A1KDM4ENPC1
SCHEMBL24770573 0.80 KDM4E (0.35) ALDH1A1KDM4ECYP3A4CYP2C19CNR1
SCHEMBL17321052 0.79 KCNJ6 (0.39) ALDH1A1KDM4EGAA
SCHEMBL9906364 0.78 CNR1 (0.43) GRNSORT1ALDH1A1KDM4ENPC1
SCHEMBL12859076 0.77 MAPK14 (0.41) MAPK14GRNSORT1ALDH1A1KDM4E
SCHEMBL12789841 0.77 GRN (0.36) GRNSORT1ALDH1A1KDM4ENPC1
SCHEMBL15898809 0.77 MAPK1 (0.34) CNR1CNR2MAPK1
SCHEMBL13114437 0.77 CNR1 (0.41) MAPK14GRNSORT1ALDH1A1KDM4E
SCHEMBL15069908 0.76 KDM4E (0.42) MAPK14GRNSORT1ALDH1A1KDM4E
SCHEMBL12789852 0.75 GRN (0.35) GRNSORT1ALDH1A1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8198308-B2 Chemical compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-12 US disclosed
US-20110059938-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-03-10 US disclosed
US-20080182837-A1 NEW CHEMICAL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-07-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110059938-A1 NEW CHEMICAL COMPOUNDS CCNA1, CCNT1, MKI67 MAPK14 2013/4885GRN 1532/4885SORT1 3054/4885
US-20080182837-A1 NEW CHEMICAL COMPOUNDS CCNA1, CCNT1, MKI67 MAPK14 2013/4885GRN 1532/4885SORT1 3054/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.