SCHEMBL9911316

SCHEMBL9911316

CC(=O)OC[C@@H]1CCC(OC(C)=O)O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.40
CYP3A4 P08684 3/20 0.38
CYP2D6 P10635 2/20 0.38
THRB P10828 2/20 0.38
CYP2C19 P33261 2/20 0.38
CYP2C9 P11712 1/20 0.38
HSD17B10 Q99714 2/20 0.37
PDK1 Q15118 1/20 0.37
NR3C1 P04150 1/20 0.36
FYN P06241 1/20 0.36
ADRA2A P08913 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
ADRA2B P18089 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
ALDH1A1 P00352 3/20 0.36
CA12 O43570 6/20 0.35
CA1 P00915 6/20 0.35
CA2 P00918 6/20 0.35
CA9 Q16790 6/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6981519 1.00 TSHR (0.40) TSHRCYP3A4CYP2D6THRBCYP2C19
SCHEMBL19060085 1.00 TSHR (0.40) TSHRCYP3A4CYP2D6THRBCYP2C19
SCHEMBL24632392 1.00 TSHR (0.40) TSHRCYP3A4CYP2D6THRBCYP2C19
SCHEMBL27413998 1.00 TSHR (0.40) TSHRCYP3A4CYP2D6THRBCYP2C19
SCHEMBL29014344 0.90 TSHR (0.38) TSHRCYP3A4CYP2D6THRBCYP2C19
SCHEMBL14277080 0.86 TSHR (0.40) TSHRCYP3A4CYP2D6THRBCYP2C19
SCHEMBL6935885 0.86 PDK1 (0.37) TSHRCYP3A4CYP2D6THRBCYP2C19
SCHEMBL20776380 0.82 PDK1 (0.34) CYP3A4CYP2D6THRBCYP2C19CYP2C9
SCHEMBL21728835 0.82 PDK1 (0.34) CYP3A4CYP2D6THRBCYP2C19CYP2C9
SCHEMBL17831609 0.81 TSHR (0.42) TSHRCYP2D6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3854799-B1 CYCLIC DINUCLEOTIDE ANALOGUE, PHARMACEUTICAL COMPOSITION THEREOF, AND APPLICATION SHANGHAI DE NOVO PHARMATECH CO LTD (CN) 2024-07-17 EP disclosed
WO-2023147161-A2 NICOTINATE AND NICOTINAMIDE RIBOSIDE-BASED COMPOUNDS AND DERIVATIVES THEREOF New Frontier Bio, Inc. (US) 2023-08-03 WO disclosed
WO-2021108291-A1 SYNTHESIS OF 3'-RNA OLIGONUCLEOTIDES ALNYLAM PHARMACEUTICALS, INC. (US) 2021-06-03 WO disclosed
US-20200397807-A1 NICOTINYL RIBOSIDE COMPOUNDS AND THEIR USES MITOPOWER LLC 2020-12-24 US disclosed
US-8193342-B2 Method for preparing furanose compounds ANADYS PHARMACEUTICALS, INC. (US) 2012-06-05 US disclosed
US-20110275589-A1 3,5-DISUBSTITUTED AND 3,5,7-TRISUBSTITUTED-3H-OXAZOLO AND 3H-THIAZOLO[4,5-d]PYRIMIDIN-2-ONE COMPOUNDS AND PRODRUGS THEREOF ANADYS PHARMACEUTICALS, INC. (US) 2011-11-10 US disclosed
US-20110172447-A1 METHOD FOR PREPARING FURANOSE COMPOUNDS ANADYS PHARMACEUTICALS, INC. (US) 2011-07-14 US disclosed
US-7928085-B2 P-toluene sulfonic acid salt of 5-amino-3-(2′-O-acetyl-3′-deoxy-β-D-ribofuranosyl)-3H-thiazole[4,5-d]pyrimidine-2-one and methods for preparation ANADYS PHARMACEUTICALS, INC. (US) 2011-04-19 US disclosed
US-20090197826-A1 P-Toluene Sulfonic Acid Salt of 5-Amino-3-(2'-O-Acetyl-3'-Deoxy-Beta-D-Ribofuranosyl)-3H-Thiazole[4,5-d]pyrimidine-2-one and Methods for Preparation ANADYS PHARMACEUTICALS, INC. (US) 2009-08-06 US disclosed
US-7560544-B2 Immunomodulators; hepatitis C virus; 5-amino-3-(O-D-ribofuranosylthiazolo[4,5-d]pyrimidine-2,7(3H,6H) dione (7-thia-8-oxoguanosine) ANADYS PHARMACEUTICALS, INC. (US) 2009-07-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200397807-A1 NICOTINYL RIBOSIDE COMPOUNDS AND THEIR USES NADK, NNT, NAMPT TSHR 3343/4885CYP3A4 1369/4885CYP2D6 1473/4885
US-20090197826-A1 P-Toluene Sulfonic Acid Salt of 5-Amino-3-(2'-O-Acetyl-3'-Deoxy-Beta-D-Ribofuranosyl)-3H-Thiazole[4,5-d]pyrimidine-2-one and Methods for Preparation DPYD, APRT, TYMS TSHR 2466/4885CYP3A4 2343/4885CYP2D6 1030/4885
US-20110275589-A1 3,5-DISUBSTITUTED AND 3,5,7-TRISUBSTITUTED-3H-OXAZOLO AND 3H-THIAZOLO[4,5-d]PYRIMIDIN-2-ONE COMPOUNDS AND PRODRUGS THEREOF TLR5, THPO, IDO1 TSHR 2594/4885CYP3A4 181/4885CYP2D6 123/4885
US-20110172447-A1 METHOD FOR PREPARING FURANOSE COMPOUNDS DPYD, TYMS, TST TSHR 3132/4885CYP3A4 859/4885CYP2D6 231/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.