SCHEMBL9911547

SCHEMBL9911547

CC(C)C(=O)Cc1c(Cl)cccc1Cl

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.59
KMT2A Q03164 4/20 0.49
ADRA2A P08913 2/20 0.49
MEN1 O00255 2/20 0.49
LMNA P02545 1/20 0.49
CYP3A4 P08684 1/20 0.49
HTR1A P08908 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
MAOA P21397 1/20 0.49
ADRA1D P25100 1/20 0.49
HTR2A P28223 1/20 0.49
HTR2C P28335 1/20 0.49
MAPK1 P28482 1/20 0.49
CYP2C19 P33261 1/20 0.49
ADRA1A P35348 1/20 0.49
DRD3 P35462 1/20 0.49
OPRK1 P41145 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1401627 0.83 AKR1B1 (0.58) AKR1B1KMT2AADRA2AMEN1LMNA
SCHEMBL9911546 0.80 CTBP2 (0.51) KMT2ALMNAMAPK1MAPTALDH1A1
SCHEMBL11243678 0.79 AKR1B1 (0.68) AKR1B1KMT2AADRA2AMEN1LMNA
SCHEMBL2421854 0.77 AKR1B1 (0.65) AKR1B1KMT2AADRA2AMEN1LMNA
SCHEMBL2525484 0.74 AKR1B1 (0.68) AKR1B1KMT2AADRA2AMEN1LMNA
SCHEMBL109215 0.74 AKR1B1 (1.00) AKR1B1KMT2AADRA2AMEN1LMNA
SCHEMBL7644229 0.73 AKR1B1 (0.50) AKR1B1KMT2AADRA2AMEN1LMNA
SCHEMBL4685080 0.72 AKR1B1 (0.65) AKR1B1KMT2AADRA2AMEN1LMNA
SCHEMBL9272252 0.72 AKR1B1 (0.65) AKR1B1KMT2AADRA2AMEN1LMNA
Hydrochloric Acid SCHEMBL1374156 0.72 AKR1B1 (0.95) AKR1B1KMT2AADRA2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8198458-B2 Non-nucleoside reverse transcriptase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-12 US disclosed
US-7517998-B2 Benzothiazole or benzothiazine derivative of dipyrido(2,3;b:2',3'-e) diazepin-6-one; viricide against human t-cell leukemia/lymphoma virus BOEHRINGER INGELHEIM INTERNATIONAL GMBH 2009-04-14 US disclosed
US-7517998-B2 Benzothiazole or benzothiazine derivative of dipyrido(2,3;b:2',3'-e) diazepin-6-one; viricide against human t-cell leukemia/lymphoma virus BOEHRINGER INGELHEIM INTERNATIONAL GMBH 2009-04-14 US disclosed