SCHEMBL9912411

SCHEMBL9912411

Cc1ccc(-c2c(C)cnn2C)c(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 6/20 0.47
HSD11B1 P28845 2/20 0.38
DRD1 P21728 1/20 0.38
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
TP53 P04637 1/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
BRD4 O60885 2/20 0.35
CRHR1 P34998 3/20 0.35
KAT2B Q92831 1/20 0.34
BRD9 Q9H8M2 1/20 0.34
NR3C1 P04150 1/20 0.34
KCNH2 Q12809 1/20 0.33
HIF1A Q16665 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14996668 0.87 HSD11B1 (0.53) PDE2AHSD11B1CRHR1KCNH2
SCHEMBL859493 0.84 PDE2A (0.46) PDE2AHSD11B1
SCHEMBL13076121 0.80 PDE2A (0.43) PDE2AHSD11B1NPC1RAB9ATP53
SCHEMBL14996545 0.80 PDE2A (0.43) PDE2AHSD11B1
SCHEMBL13076118 0.79 PDE2A (0.43) PDE2AHSD11B1NPC1RAB9ATP53
SCHEMBL859848 0.77 PDE2A (0.41) PDE2AHSD11B1NPC1RAB9ATP53
SCHEMBL846412 0.73 GRK6 (0.40) PDE2AHPGDTSHR
SCHEMBL9911401 0.71 ALDH1A1 (0.54) PDE2AHSD11B1DRD1NPC1RAB9A
SCHEMBL11507014 0.71 NPC1 (0.46) HSD11B1NPC1RAB9ATP53HPGD
SCHEMBL14996666 0.71 PDE2A (0.41) PDE2ANPC1RAB9ATDP1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8198458-B2 Non-nucleoside reverse transcriptase inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-12 US disclosed
US-7517998-B2 Benzothiazole or benzothiazine derivative of dipyrido(2,3;b:2',3'-e) diazepin-6-one; viricide against human t-cell leukemia/lymphoma virus BOEHRINGER INGELHEIM INTERNATIONAL GMBH 2009-04-14 US disclosed