SCHEMBL9917

SCHEMBL9917

Cc1noc(-c2ccccc2-c2ccc(C3(C(=O)O)CC3)cc2)c1CN1C(=O)OC[C@@H]1c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SCD5 Q86SK9 1/20 0.43
ABCC3 O15438 1/20 0.40
ABCC4 O15439 1/20 0.40
ABCB11 O95342 1/20 0.40
CYP2C8 P10632 1/20 0.40
CYP2C9 P11712 1/20 0.40
ABCB4 P21439 1/20 0.40
LPAR1 Q92633 1/20 0.40
ABCC2 Q92887 1/20 0.40
SLCO1B3 Q9NPD5 1/20 0.40
SLCO1B1 Q9Y6L6 1/20 0.40
HDAC1 Q13547 2/20 0.37
TAS2R8 Q9NYW2 2/20 0.36
GLS O94925 4/20 0.33
PTGDR2 Q9Y5Y4 2/20 0.33
BRD4 O60885 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14779471 0.92 SCD5 (0.45) SCD5ABCC3ABCC4ABCB11CYP2C8
SCHEMBL3309 0.92 SCD5 (0.45) SCD5ABCC3ABCC4ABCB11CYP2C8
SCHEMBL9916 0.92 SCD5 (0.42) SCD5ABCC3ABCC4ABCB11CYP2C8
SCHEMBL9915 0.92 SCD5 (0.42) SCD5ABCC3ABCC4ABCB11CYP2C8
SCHEMBL10039 0.87 HDAC1 (0.39) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL14778153 0.85 SCD5 (0.42) SCD5ABCC3ABCC4ABCB11CYP2C8
SCHEMBL3778 0.85 SCD5 (0.42) SCD5ABCC3ABCC4ABCB11CYP2C8
SCHEMBL9419 0.82 CYP2C9 (0.40) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL10037 0.79 HDAC1 (0.40) ABCC3ABCC4ABCB11CYP2C8CYP2C9
SCHEMBL10038 0.79 HDAC1 (0.40) ABCC3ABCC4ABCB11CYP2C8CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2483251-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-08-08 EP disclosed
WO-2011041462-A2 POLYCYCLIC COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-04-07 WO disclosed