SCHEMBL9924168

SCHEMBL9924168

Cc1cc(C(=O)N[C@H]2CC[C@H](N/C(=N\C(=O)c3ccc(F)c(F)c3)Nc3cccc(Cl)c3)CC2)ccn1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 3/20 0.44
AR P10275 3/20 0.43
MCHR1 Q99705 5/20 0.42
GRM5 P41594 1/20 0.41
MAPK11 Q15759 1/20 0.40
MAPK14 Q16539 1/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
CRHR1 P34998 1/20 0.40
BRAF P15056 1/20 0.40
NUDT1 P36639 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9924169 0.86 CRHR1 (0.49) GRM5L3MBTL1CRHR1
SCHEMBL9924422 0.84 KCNQ3 (0.42) MCHR1GRM5MAPT
SCHEMBL17206698 0.83 GRM5 (0.51) ACKR3GRM5MAPT
SCHEMBL9924260 0.83 MEN1 (0.46) ACKR3MAPTL3MBTL1CRHR1
SCHEMBL17206628 0.82 MEN1 (0.45) ACKR3MAPTCRHR1
SCHEMBL17206687 0.82 KCNQ3 (0.45) ARGRM5MAPTBRAF
SCHEMBL9924424 0.81 TRPV1 (0.45) ACKR3MAPT
SCHEMBL9924144 0.81 MEN1 (0.42) MAPT
SCHEMBL9924171 0.80 DRD2 (0.47) MAPT
SCHEMBL9924128 0.79 MEN1 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9169199-B2 Cycloalkyl guanidine F1F0-ATPase inhibitors and therapeutic uses thereof LYCERA CORPORATION (US) 2015-10-27 US disclosed
WO-2012078867-A2 CYCLOALKYL GUANIDINE F1F0-ATPASE INHIBITORS AND THERAPEUTIC USES THEREOF LYCERA CORPORATION (US) 2012-06-14 WO disclosed