SCHEMBL9924385

SCHEMBL9924385

O=c1[nH]cnc2ccc(Cc3cnc4ccc(-c5ccccc5)nn34)cc12

nearest known ligand 0.72

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MET P08581 7/20 0.72
IP6K1 Q92551 6/20 0.51
IP6K3 Q96PC2 3/20 0.51
IP6K2 Q9UHH9 3/20 0.51
PRMT5 O14744 1/20 0.44
WDR77 Q9BQA1 1/20 0.44
FYN P06241 3/20 0.43
PIK3CD O00329 1/20 0.43
ACVR1 Q04771 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2697213 0.84 MET (1.00) METIP6K1IP6K3IP6K2
SCHEMBL9924372 0.79 MET (0.68) METFYN
SCHEMBL2493581 0.77 MET (0.82) MET
SCHEMBL1656793 0.76 MET (0.74) MET
SCHEMBL9924374 0.74 MET (0.56) METFYN
SCHEMBL9924368 0.74 MET (0.73) METFYN
SCHEMBL9924380 0.73 FYN (0.56) METFYN
SCHEMBL9924377 0.73 MET (0.63) METFYN
SCHEMBL9924378 0.72 FYN (0.51) METFYN
SCHEMBL9924390 0.72 FYN (0.52) METFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130303529-A1 FUSED HETEROCYCLIC DERIVATIVES AND METHODS OF USE AMGEN INC (US) 2013-11-14 US disclosed
US-8524900-B2 Fused heterocyclic derivatives and methods of use AMGEN INC. (US) 2013-09-03 US disclosed
US-20120148531-A1 FUSED HETEROCYCLIC DERIVATIVES AND METHODS OF USE AMGEN INC. (US) 2012-06-14 US disclosed
US-20120107275-A1 FUSED HETEROCYCLIC DERIVATIVES AND METHODS OF USE AMGEN INC. (US) 2012-05-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120148531-A1 FUSED HETEROCYCLIC DERIVATIVES AND METHODS OF USE HGF, HGFAC, MET MET 3/4885IP6K1 3165/4885IP6K3 3105/4885
US-20130303529-A1 FUSED HETEROCYCLIC DERIVATIVES AND METHODS OF USE HGF, HGFAC, MET MET 3/4885IP6K1 3165/4885IP6K3 3105/4885
US-20120107275-A1 FUSED HETEROCYCLIC DERIVATIVES AND METHODS OF USE HGF, HGFAC, MET MET 3/4885IP6K1 3165/4885IP6K3 3105/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.