SCHEMBL9925362

SCHEMBL9925362

C#C/C(N)=N\C(=O)c1cc(C)c2nccc(-c3c(Cl)cccc3Cl)c2c1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR5A P47898 8/20 0.38
PTGDR2 Q9Y5Y4 4/20 0.38
CYP2C9 P11712 1/20 0.35
PTGS1 P23219 1/20 0.35
SLC6A4 P31645 1/20 0.35
CYP2C19 P33261 1/20 0.35
PTGS2 P35354 1/20 0.35
HTR7 P34969 4/20 0.34
HTR2B P41595 4/20 0.34
DYRK1A Q13627 1/20 0.32
PIK3R2 O00459 1/20 0.31
MAPK1 P28482 2/20 0.31
MAPK3 P27361 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9907837 0.89 HTR5A (0.47) HTR5APTGDR2HTR7HTR2B
SCHEMBL12875077 0.89 HTR5A (0.45) HTR5APTGDR2CYP2C9PTGS1SLC6A4
SCHEMBL12874635 0.87 HTR5A (0.41) HTR5APTGDR2
SCHEMBL15500584 0.86 PTGDR2 (0.35) HTR5APTGDR2CYP2C9PTGS1SLC6A4
SCHEMBL12875043 0.85 HTR5A (0.45) HTR5APTGDR2CYP2C9PTGS1SLC6A4
SCHEMBL12874645 0.84 HTR5A (0.38) HTR5A
SCHEMBL9907822 0.83 HTR5A (0.55) HTR5APTGDR2HTR7HTR2B
SCHEMBL12874648 0.83 CDC7 (0.37) HTR5APTGDR2CYP2C9CYP2C19
SCHEMBL12874646 0.82 GRM2 (0.36) HTR5AMAPK1
SCHEMBL9907464 0.80 PTGDR2 (0.46) PTGDR2CYP2C9PTGS1SLC6A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2463276-A1 NITROGENOUS-RING ACYLGUANIDINE DERIVATIVE Astellas Pharma Inc. (JP) 2012-06-13 EP disclosed