SCHEMBL9925422

SCHEMBL9925422

N#Cc1ccc(-c2c(Cl)cnc3ccc(C(=O)N=O)cc23)c(F)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR5A P47898 8/20 0.60
TNF P01375 1/20 0.35
SLC22A12 Q96S37 2/20 0.34
S1PR3 Q99500 2/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
MTOR P42345 1/20 0.34
PIK3CG P48736 1/20 0.34
PRKDC P78527 1/20 0.34
ATM Q13315 1/20 0.34
ATR Q13535 1/20 0.34
MAP3K8 P41279 1/20 0.34
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9909288 0.89 HTR5A (0.77) HTR5APIK3CAPIK3CBMTORPIK3CG
SCHEMBL9909253 0.89 HTR5A (0.55) HTR5ATNFSLC22A12S1PR3PIK3CA
SCHEMBL12875061 0.86 HTR5A (0.64) HTR5ATNFPIK3CAPIK3CBMTOR
SCHEMBL9925448 0.85 HTR5A (0.52) HTR5ATNFPIK3CAPIK3CBMTOR
SCHEMBL9909242 0.75 HTR5A (0.59) HTR5APIK3CAPIK3CBMTORPIK3CG
SCHEMBL9907842 0.75 HTR5A (1.00) HTR5A
SCHEMBL9907497 0.74 HTR5A (0.72) HTR5A
SCHEMBL9909265 0.73 PDE5A (0.42) HTR5ASLC22A12EGLN1
SCHEMBL9907888 0.73 HTR5A (0.81) HTR5A
SCHEMBL9925369 0.73 HTR5A (0.48) HTR5AHDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2463276-A1 NITROGENOUS-RING ACYLGUANIDINE DERIVATIVE Astellas Pharma Inc. (JP) 2012-06-13 EP disclosed