SCHEMBL9925842

SCHEMBL9925842

CC(O)[C@H](NC(=O)c1ccc(F)c(Br)c1)C(=O)NO

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.43
CA1 P00915 2/20 0.43
ANPEP P15144 2/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
PPARG P37231 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL402028 1.00 CA2 (0.43) CA2CA1ANPEPPDE4APDE4B
SCHEMBL405477 0.89 CCR1 (0.47) ANPEPPDE4APDE4BPDE4CPDE4D
SCHEMBL402851 0.89 CCR1 (0.47) ANPEPPDE4APDE4BPDE4CPDE4D
SCHEMBL2873360 0.88 CA2 (0.56) CA2CA1ALDH1A1GAAPKM
SCHEMBL403937 0.85 TAS1R3 (0.51) CA2CA1ALDH1A1GAAPKM
SCHEMBL9902468 0.85 TAS1R3 (0.51) CA2CA1ALDH1A1GAAPKM
SCHEMBL1109256 0.85 TAS1R3 (0.51) CA2CA1ALDH1A1GAAPKM
SCHEMBL12055901 0.85 NPC1 (0.48) CA2CA1ALDH1A1
SCHEMBL12837671 0.83 CA2 (0.43) CA2CA1HDAC6ALDH1A1GAA
SCHEMBL403958 0.83 HDAC8 (0.55) ANPEPPDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1618087-B1 ANTIBACTERIAL AGENTS NOVARTIS VACCINES & DIAGNOSTIC (US) 2012-06-13 EP disclosed