SCHEMBL9925877

SCHEMBL9925877

C=C(N[C@@H](CN)C(=O)NO)c1ccc(-c2cccc([N+](=O)[O-])c2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.43
MMP9 P14780 2/20 0.43
MMP8 P22894 1/20 0.43
HDAC2 Q92769 1/20 0.43
MME P08473 1/20 0.43
PLG P00747 1/20 0.41
PLAU P00749 1/20 0.41
PLAT P00750 1/20 0.41
ABCB1 P08183 2/20 0.40
ALDH1A1 P00352 2/20 0.40
KDM4E B2RXH2 1/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
CNR1 P21554 1/20 0.40
SLC6A4 P31645 1/20 0.39
NQO2 P16083 1/20 0.39
ALOX5 P09917 1/20 0.39
MMP1 P03956 1/20 0.39
TRPM2 O94759 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14224159 0.89 HDAC2 (0.50) MMP2MMP9MMP8HDAC2MME
SCHEMBL399936 0.75 FFAR1 (0.44) ALDH1A1MAPT
SCHEMBL404504 0.75 FFAR1 (0.44) ALDH1A1MAPT
SCHEMBL5944081 0.74 HDAC2 (0.59) MMP2MMP9MMP8HDAC2PLG
SCHEMBL403123 0.72 HTT (0.47) MMP2MMP9MMP8HDAC2PLG
SCHEMBL27889371 0.71 TSHR (0.68) MMP2MMP9MMP8HDAC2PLG
SCHEMBL1109277 0.71 HPGDS (0.65)
SCHEMBL1109563 0.71 HPGDS (0.49) MMEALDH1A1MAPT
SCHEMBL1109400 0.70 CTSB (0.47)
SCHEMBL3765312 0.70 TP53 (0.67) MMP2MMP9MMP8HDAC2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1618087-B1 ANTIBACTERIAL AGENTS NOVARTIS VACCINES & DIAGNOSTIC (US) 2012-06-13 EP disclosed