SCHEMBL9926046

SCHEMBL9926046

Cc1ccc(C)c(N2CCN(C(=O)[C@@H]3CN(S(=O)(=O)c4ccc(Cl)cc4)C[C@H]3c3ccccc3)CC2)c1

nearest known ligand 0.52

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MC4R P32245 12/20 0.52
AR P10275 5/20 0.49
USP2 O75604 1/20 0.48
HTT P42858 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
LMNA P02545 1/20 0.48
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5264649 1.00 MC4R (0.52) MC4RARUSP2HTTNPSR1
SCHEMBL9926039 0.91 LMNA (0.52) MC4RARUSP2HTTNPSR1
SCHEMBL9926136 0.86 USP2 (0.57) ARUSP2HTTNPSR1LMNA
SCHEMBL14269767 0.86 USP2 (0.57) ARUSP2HTTNPSR1LMNA
SCHEMBL9926098 0.86 USP2 (0.57) ARUSP2HTTNPSR1LMNA
SCHEMBL9926101 0.85 SMN1; SMN2 (0.47) MC4RARUSP2LMNAMAPT
SCHEMBL4849442 0.85 LMNA (0.48) ARUSP2HTTLMNAMAPT
SCHEMBL4847578 0.85 LMNA (0.48) ARUSP2HTTLMNAMAPT
SCHEMBL9925998 0.85 AR (0.46) MC4RARUSP2MAPT
SCHEMBL5270813 0.85 AR (0.46) MC4RARUSP2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1836180-B1 SULFONYL PYRROLIDINES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS DRUGS SANOFI SA (FR) 2012-06-13 EP disclosed
US-7468369-B2 Sulfonyl pyrrolidines, method for producing the same and their use as drugs SANOFI-AVENTIS (FR) 2008-12-23 US disclosed
US-20080045540-A1 SULFONYL PYRROLIDINES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS DRUGS SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2008-02-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080045540-A1 SULFONYL PYRROLIDINES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS DRUGS SLC5A1, SLC5A2, KCNJ1 MC4R 1509/4885AR 4287/4885USP2 3511/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.