SCHEMBL9926495

SCHEMBL9926495

O=C/C=C1/C(=O)Nc2cccc(O)c21

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 2/20 0.58
PLK4 O00444 3/20 0.45
PLK1 P53350 3/20 0.45
TGM2 P21980 6/20 0.43
EPHX2 P34913 1/20 0.40
MAP3K7 O43318 1/20 0.39
TAB1 Q15750 1/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
MAPK1 P28482 1/20 0.39
RET P07949 2/20 0.39
FLT3 P36888 1/20 0.39
PDGFRB P09619 1/20 0.39
CES1 P23141 1/20 0.39
KDR P35968 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2331366 0.78 PDPK1 (0.54) PDPK1PLK4PLK1TGM2ALDH1A1
SCHEMBL5728638 0.74 PDPK1 (1.00) PDPK1RETFLT3PDGFRBKDR
SCHEMBL27553562 0.74 TGM2 (0.73) PDPK1TGM2MAP3K7TAB1
SCHEMBL5728634 0.74 PDPK1 (1.00) PDPK1RETFLT3PDGFRBKDR
SCHEMBL6917819 0.72 PDPK1 (0.49) PDPK1PLK4PLK1TGM2ALDH1A1
SCHEMBL21837129 0.72 EPHX2 (0.65) PDPK1PLK4PLK1TGM2EPHX2
SCHEMBL4861892 0.64 KDR (0.60) PDPK1TGM2EPHX2ALDH1A1MAPT
SCHEMBL4996116 0.64 TGM2 (0.48) PDPK1TGM2ALDH1A1MAPTNPSR1
SCHEMBL4996113 0.64 TGM2 (0.48) PDPK1TGM2ALDH1A1MAPTNPSR1
SCHEMBL4861881 0.64 KDR (0.60) PDPK1TGM2EPHX2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012078519-A2 3-ACYLIDENE-2-OXOINDOLE DERIVATIVES FOR INHIBITION OF TRANSGLUTAMINASE 2 NUMERATE, INC. (US) 2012-06-14 WO disclosed