Brivudine

Brivudine

SCHEMBL99350

O=c1[nH]c(=O)n([C@H]2C[C@H](O)[C@@H](CO)O2)cc1/C=C/Br

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TK1 P04183 4/20 1.00
CYP1A2 P05177 1/20 1.00
CYP3A4 P08684 1/20 1.00
TSHR P16473 1/20 1.00
BLM P54132 1/20 1.00
PMP22 Q01453 1/20 1.00
NPSR1 Q6W5P4 1/20 1.00
LMNA P02545 2/20 0.66
SMN1; SMN2 Q16637 2/20 0.66
TK2 O00142 5/20 0.65
ALOX12 P18054 1/20 0.62
ADRA1A P35348 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Brivudine SCHEMBL13030272 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL4283383 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL4314668 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL141407 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL13674189 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL1172398 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL4283382 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL5983819 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL21316784 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM
Brivudine SCHEMBL15405329 1.00 TK1 (1.00) TK1CYP1A2CYP3A4TSHRBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 5066 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260144879-A1 ANTI-VIRAL AND HEPATIC-TARGETED DRUGS AI-BIOPHARMA (FR) 2026-05-28 US claimed
WO-2026107113-A1 MODIFIED CELLS FOR PROGRAMMING EXTRA ENVELOPED VIRUSES (EEVs) AND THEIR USE FOR PRODUCING THE EEVs, THE PROGRAMMED EEVs AND USES THEREOF CALIDI BIOTHERAPEUTICS (NEVADA), INC. (US) 2026-05-21 WO claimed
CN-122056884-A Methods of treating pancreatic cancer 坎莫森特里克斯公司 2026-05-19 CN claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
EP-3790536-B1 NANOCONTAINERS FOR TRANSPORTING NONPOLAR, LIPOPHILIC SUBSTANCES SUCH AS ANTIBIOTICS KARLSRUHER INST TECHNOLOGIE (DE) 2026-04-22 EP claimed
US-12599644-B2 Treatment of coronavirus infection with Flt3 receptor interacting lectin (FRIL) ACADEMIA SINICA (TW) 2026-04-14 US claimed
US-20260092059-A1 Broad Spectrum Antiviral Compositions and Methods EVRYS BIO, LLC (US) 2026-04-02 US claimed
US-12582148-B2 Compositions and methods for improving quality of life in patients with autism spectrum disorder FLAASK, LLC (US) 2026-03-24 US claimed
US-12576124-B2 Formulation of a conjugate of a tubulysin analog to a cell-binding molecule HANGZHOU DAC BIOTECH CO., LTD (CN) 2026-03-17 US claimed
WO-1995012313-A1 VIRUS ASSOCIATED MULTIPLE SCLEROSIS: TREATMENTS, PREVENTION AND DIAGNOSIS THEREOF PATHOGENESIS CORPORATION (US) 1995-05-11 WO claimed
WO-1994026273-A1 ACYCLOVIR DERIVATIVES FOR TOPICAL USE HOSTETLER KARL Y (US) 1994-11-24 WO claimed
US-5159067-A 5'-Diphosphohexose nucleoside pharmaceutical compositions UNIVERSITY OF GEORGIA RESEARCH FOUNDATION INC. (US) 1992-10-27 US claimed
EP-0283065-B1 COMBINATIONS OF FU AND BVU AS ANTI-ADENOCARCINOMA AGENTS Stichting REGA V.Z.W. (BE) 1991-05-29 EP claimed
US-4988678-A Fluorouracil and tetrahydrofuryl-5-fluorouracil as an antitumor agent and bromovinyluracil and 5-(2-bromovinyl-2'-deoxyuridine STICHTING REGA VZW (BE) 1991-01-29 US claimed
US-4894365-A 5-FLUOROURACIL AND BROMOVINYLURACIL STICHTING REGA VZW (BE) 1990-01-16 US claimed
EP-0143987-B1 THERAPEUTIC COMPOSITIONS ENDOWED WITH ANTIVIRAL ACTIVITY Stendardi, Anna Gioia (IT) 1989-02-22 EP claimed
EP-0143987-A1 Therapeutic compositions endowed with antiviral activity Stendardi, Anna Gioia (IT) 1985-06-12 EP claimed
EP-0090837-A1 METHOD AND COMPOSITION FOR TREATING A PATIENT SUFFERING FROM INTERFERONSUSCEPTIBLE DISORDER BERG, Kurt Frimann (DK) 1983-10-12 EP claimed
WO-1983001198-A1 METHOD AND COMPOSITION FOR TREATING A PATIENT SUFFERING FROM INTERFERON-SUSCEPTIBLE DISORDER BERG, KURT, FRIMANN 1983-04-14 WO claimed