SCHEMBL9939475

SCHEMBL9939475

Cc1noc(-c2ccc(-c3ccc(C4(C(=O)O)CC4)cc3)cc2)c1C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LPAR1 Q92633 8/20 0.54
CYP2C9 P11712 3/20 0.54
ABCC3 O15438 1/20 0.54
ABCC4 O15439 1/20 0.54
ABCB11 O95342 1/20 0.54
CYP2C8 P10632 1/20 0.54
ABCB4 P21439 1/20 0.54
ABCC2 Q92887 1/20 0.54
SLCO1B3 Q9NPD5 1/20 0.54
SLCO1B1 Q9Y6L6 1/20 0.54
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
AKR1C1 Q04828 2/20 0.39
AKR1B10 O60218 1/20 0.39
AKR1C4 P17516 1/20 0.39
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
IP6K1 Q92551 2/20 0.38
IP6K3 Q96PC2 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14794645 0.99 LPAR1 (0.53) LPAR1CYP2C9ABCC3ABCC4ABCB11
SCHEMBL14794646 0.86 LPAR1 (0.47) LPAR1CYP2C9ABCC3ABCC4ABCB11
SCHEMBL342705 0.86 OPRM1 (0.45) LPAR1CYP2C9ABCC3ABCC4ABCB11
SCHEMBL12973618 0.86 LPAR1 (0.52) LPAR1CYP2C9ABCC3ABCC4ABCB11
SCHEMBL9939476 0.84 LPAR1 (0.54) LPAR1CYP2C9ABCC3ABCC4ABCB11
SCHEMBL14711012 0.83 AKR1C3 (0.42) LPAR1CYP2C9ABCC3ABCC4ABCB11
SCHEMBL343870 0.83 ABCC3 (0.43) LPAR1CYP2C9ABCC3ABCC4ABCB11
SCHEMBL14711260 0.82 PTGS1 (0.50) LPAR1CYP2C9ABCC3ABCC4ABCB11
SCHEMBL18597706 0.82 LPAR1 (0.63) LPAR1CYP2C9ABCC3ABCC4ABCB11
SCHEMBL6674 0.82 LPAR1 (0.53) LPAR1CYP2C9ABCC3ABCC4ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012078805-A1 POLYCYCLIC LPA1 ANTAGONIST AND USES THEREOF AMIRA PHARMACEUTICALS, INC. (US) 2012-06-14 WO disclosed