SCHEMBL9940458

SCHEMBL9940458

CC1(C)OB(c2cn(C(c3ccccc3)(c3ccccc3)c3ccccc3)c3ncc(F)cc23)OC1(C)C

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 7/20 0.35
JAK2 O60674 2/20 0.31
BTK Q06187 2/20 0.31
IDO1 P14902 1/20 0.31
TDO2 P48775 1/20 0.31
HTR3A P46098 1/20 0.30
LPL P06858 1/20 0.30
LIPG Q9Y5X9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21820978 0.80 LIPE (0.33) LIPELPLLIPG
SCHEMBL9940965 0.78 LIPE (0.31) LIPEIDO1TDO2LPLLIPG
SCHEMBL16884162 0.77 LPL (0.33) LIPEJAK2BTKIDO1TDO2
SCHEMBL21821014 0.76 IRAK4 (0.32) LIPELPLLIPG
SCHEMBL30387520 0.76 IRAK4 (0.32) LIPELPLLIPG
SCHEMBL25596649 0.76 BRD4 (0.41) LIPEIDO1TDO2
SCHEMBL21820843 0.76 LIPE (0.33) LIPELPLLIPG
SCHEMBL21820851 0.75 LPL (0.33) LIPELPLLIPG
SCHEMBL24710404 0.75 CCND1 (0.35) LPLLIPG
SCHEMBL21821115 0.74 IRAK4 (0.32) LIPELPLLIPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2651940-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION Vertex Pharmaceuticals Incorporated (US) 2013-10-23 EP disclosed
WO-2012083117-A1 INHIBITORS OF INFLUENZA VIRUSES REPLICATION VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-06-21 WO disclosed