SCHEMBL9940541

SCHEMBL9940541

CC[Si](CC)(CC)CCOCn1cc(C(F)(F)F)nc1-c1cnc(Cl)cc1C

nearest known ligand 0.48

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 9/20 0.48
S1PR2 O95136 1/20 0.32
PTGS1 P23219 2/20 0.31
PTGS2 P35354 2/20 0.31
METAP2 P50579 1/20 0.31
USP1 O94782 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15282735 0.91 DGAT1 (0.60) DGAT1S1PR2PTGS1PTGS2METAP2
SCHEMBL20169338 0.85 DGAT1 (0.44) DGAT1PTGS1PTGS2METAP2
SCHEMBL15293918 0.78 DGAT1 (0.72) DGAT1
SCHEMBL18085602 0.74 DGAT1 (0.69) DGAT1PTGS1PTGS2
SCHEMBL16787746 0.73 DGAT1 (0.78) DGAT1PTGS1PTGS2USP1
SCHEMBL15293832 0.70 DGAT1 (0.64) DGAT1PTGS1PTGS2
SCHEMBL20169353 0.69 DGAT1 (0.52) DGAT1PTGS1PTGS2
SCHEMBL9940375 0.69 DGAT1 (0.61) DGAT1PTGS1PTGS2
SCHEMBL25230088 0.68 DGAT1 (0.57) DGAT1USP1
SCHEMBL9936872 0.68 DGAT1 (0.63) DGAT1PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2651915-A1 CONTINUOUS ARYCYCLIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2013-10-23 EP disclosed
WO-2012081736-A1 CONTINUOUS ARYCYCLIC COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-06-21 WO disclosed