SCHEMBL9942591

SCHEMBL9942591

Bc1cnc(-n2cccn2)c([N+](=O)[O-])c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 12/20 0.37
MEN1 O00255 8/20 0.37
MAPT P10636 8/20 0.37
KMT2A Q03164 8/20 0.37
LMNA P02545 6/20 0.37
HTT P42858 2/20 0.37
MAPK1 P28482 1/20 0.37
MDM2 Q00987 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
RAB9A P51151 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HSP90AA1 P07900 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KDM4E B2RXH2 2/20 0.33
GAA P10253 1/20 0.33
G6PD P11413 1/20 0.33
KDM4A O75164 1/20 0.32
KDM4B O94953 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1763428 0.83 ALDH1A1 (0.37) ALDH1A1MEN1MAPTKMT2ALMNA
SCHEMBL8675692 0.76 CYP1A2 (0.56) ALDH1A1MEN1MAPTKMT2ALMNA
SCHEMBL14909413 0.71 ALDH1A1 (0.40) ALDH1A1MEN1MAPTKMT2ALMNA
SCHEMBL14910448 0.71 ALDH1A1 (0.41) ALDH1A1MEN1MAPTKMT2ALMNA
SCHEMBL18983611 0.71 ALDH1A1 (0.40) ALDH1A1MEN1MAPTKMT2ALMNA
SCHEMBL14909409 0.71 ALDH1A1 (0.43) ALDH1A1MEN1MAPTKMT2ALMNA
SCHEMBL3580195 0.70 ALDH1A1 (0.40) ALDH1A1MEN1MAPTKMT2ALMNA
SCHEMBL13314707 0.69 L3MBTL1 (0.40) ALDH1A1MEN1MAPTKMT2ALMNA
SCHEMBL13310611 0.69 ALDH1A1 (0.52) ALDH1A1MEN1MAPTKMT2ALMNA
SCHEMBL30888284 0.69 ALDH1A1 (0.52) ALDH1A1MEN1MAPTKMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1363705-B9 COMPOSITION AND ANTIVIRAL ACTIVITY OF SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES BRISTOL MYERS SQUIBB CO (US) 2012-11-07 EP disclosed
EP-1363705-B1 COMPOSITION AND ANTIVIRAL ACTIVITY OF SUBSTITUTED AZAINDOLEOXOACETIC PIPERAZINE DERIVATIVES BRISTOL MYERS SQUIBB CO (US) 2012-06-13 EP disclosed