SCHEMBL9943564

SCHEMBL9943564

CCn1c(=O)[nH]c(N)c(NC(=O)C#C[Si](C)(C)C)c1=O

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.35
ADORA2A P29274 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
POLB P06746 1/20 0.32
MAPT P10636 1/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
ADORA2B P29275 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9904076 0.90 ADORA2B (0.37) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL9904219 0.80 EEF2K (0.34) ADORA2AMEN1KMT2AADORA2B
SCHEMBL9943417 0.70 EPHX2 (0.35) MEN1ALDH1A1KMT2A
SCHEMBL2328928 0.65 MAPT (0.47) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL1866393 0.62 ADORA2B (0.44) ADORA2AMEN1ALDH1A1KMT2ASMN1; SMN2
SCHEMBL12079923 0.61 ADORA1 (0.52) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL1944878 0.60 MAPT (0.42) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL3447830 0.59 MAPT (0.42) ADORA2APOLBMAPTMEN1ALDH1A1
SCHEMBL15780384 0.57 MAPT (0.46) PDE4AADORA2APDE4BPDE4CPDE4D
SCHEMBL7093037 0.56 MAPT (0.49) POLBMAPTMEN1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2465859-A1 8-Triazolylxanthine derivatives, processes for their production and their use as adenosine receptor antagonists Life & Brain GmbH (DE) 2012-06-20 EP disclosed