SCHEMBL9943774

SCHEMBL9943774

Nc1ncccc1-n1cnnn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.49
NPSR1 Q6W5P4 1/20 0.49
NOTUM Q6P988 3/20 0.44
KDM4E B2RXH2 2/20 0.41
KMT2A Q03164 2/20 0.41
LMNA P02545 1/20 0.40
JAK2 O60674 2/20 0.39
JAK1 P23458 2/20 0.39
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
AMY1A P0DUB6 1/20 0.38
MAPT P10636 2/20 0.38
F2 P00734 1/20 0.38
MITF O75030 1/20 0.38
GAA P10253 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TSHR P16473 1/20 0.37
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16114399 0.79 ALDH1A1 (0.49) ALDH1A1NPSR1NOTUMKDM4EKMT2A
SCHEMBL5855553 0.78 ALDH1A1 (0.45) ALDH1A1NPSR1NOTUMKDM4EKMT2A
SCHEMBL18284817 0.76 NOTUM (0.43) NOTUMNOS3NOS1NOS2AMY1A
SCHEMBL12615992 0.76 ALDH1A1 (0.68) ALDH1A1NPSR1NOTUMKDM4EKMT2A
SCHEMBL15758070 0.76 KCNJ1 (0.44) ALDH1A1NPSR1NOTUMKDM4EKMT2A
SCHEMBL30084182 0.76 ALDH1A1 (0.58) ALDH1A1NPSR1NOTUMKDM4EKMT2A
SCHEMBL5330184 0.76 ALDH1A1 (0.58) ALDH1A1NPSR1NOTUMKDM4EKMT2A
SCHEMBL17978905 0.75 ALDH1A1 (0.45) ALDH1A1NPSR1NOTUMKDM4EKMT2A
SCHEMBL5854751 0.75 ALDH1A1 (0.49) ALDH1A1NPSR1NOTUMKDM4EKMT2A
SCHEMBL11146019 0.73 ALDH1A1 (0.54) ALDH1A1NPSR1NOTUMKDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2464228-A1 SUBSTITUTED CYCLOPROPYL COMPOUNDS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT Merck Sharp & Dohme Corp. (US) 2012-06-20 EP claimed