SCHEMBL9947006

SCHEMBL9947006

CNc1cc(NCc2nccn2C)c(C(=O)NC2CCC(C(F)(F)F)CC2)cc1N

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGES O14684 8/20 0.53
TRPM5 Q9NZQ8 1/20 0.36
CD38 P28907 2/20 0.36
TYK2 P29597 3/20 0.36
IRAK4 Q9NWZ3 5/20 0.35
TTK P33981 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9946585 1.00 PTGES (0.53) PTGESTRPM5CD38TYK2IRAK4
SCHEMBL9944937 0.90 PTGES (0.43) PTGESCD38
SCHEMBL9947005 0.84 PTGES (0.52) PTGESCD38TYK2
SCHEMBL9946715 0.84 PTGES (0.52) PTGESCD38TYK2
SCHEMBL9946693 0.80 PTGES (0.46) PTGESIRAK4
SCHEMBL9947033 0.80 PTGES (0.46) PTGESIRAK4
SCHEMBL9942023 0.77 PTGES (0.47) PTGESCD38TYK2TTK
SCHEMBL11970141 0.76 HPGD (0.42) PTGES
SCHEMBL10170842 0.76 HPGD (0.42) PTGES
SCHEMBL9944936 0.76 PTGES (0.41) PTGESCD38

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076673-A1 6-AMINO-2-PHENYLAMINO-1H-BENZIMIDAZOLE-5-CARBOXAMIDE- DERIVATIVES AND THEIR USE AS MICROSOMAL PROSTAGLANDIN E2 SYNTHASE-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-14 WO disclosed