SCHEMBL9947033

SCHEMBL9947033

CNc1cc(NCCCO)c(C(=O)NC2CCC(C(F)(F)F)CC2)cc1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 6/20 0.46
HTR4 Q13639 3/20 0.35
S100A4 P26447 1/20 0.34
MAPK14 Q16539 1/20 0.34
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
IRAK4 Q9NWZ3 2/20 0.33
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA3 P07451 1/20 0.33
CA6 P23280 1/20 0.33
CA5A P35218 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
CA13 Q8N1Q1 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CA5B Q9Y2D0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9946693 1.00 PTGES (0.46) PTGESHTR4S100A4MAPK14ALDH1A1
SCHEMBL9944890 0.87 CNR2 (0.43) HTR4S100A4MAPK14CNR1CNR2
SCHEMBL10170842 0.82 HPGD (0.42) PTGESS100A4MAPK14POLBHPGD
SCHEMBL11970141 0.82 HPGD (0.42) PTGESS100A4MAPK14POLBHPGD
SCHEMBL9899306 0.80 PTGES (0.46) PTGESS100A4IRAK4HPGD
SCHEMBL9899308 0.80 PTGES (0.46) PTGESS100A4IRAK4HPGD
SCHEMBL9946585 0.80 PTGES (0.53) PTGESIRAK4
SCHEMBL9947006 0.80 PTGES (0.53) PTGESIRAK4
SCHEMBL9946720 0.76 PTGES (0.44) PTGESALDH1A1
SCHEMBL9947009 0.76 PTGES (0.48) PTGESS100A4ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076673-A1 6-AMINO-2-PHENYLAMINO-1H-BENZIMIDAZOLE-5-CARBOXAMIDE- DERIVATIVES AND THEIR USE AS MICROSOMAL PROSTAGLANDIN E2 SYNTHASE-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-14 WO disclosed