SCHEMBL9947086

SCHEMBL9947086

CNc1cc(NC)c([N+](=O)[O-])cc1C(=O)N[C@H]1CC[C@H](C(F)(F)F)CC1

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
HCAR3 P49019 2/20 0.38
MITF O75030 1/20 0.38
CDC25B P30305 1/20 0.37
POLB P06746 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
HTT P42858 1/20 0.36
HPGD P15428 2/20 0.35
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1727199 0.91 ALDH1A1 (0.45) ALDH1A1HCAR3MITFCDC25BPOLB
SCHEMBL1727200 0.91 ALDH1A1 (0.45) ALDH1A1HCAR3MITFCDC25BPOLB
SCHEMBL9897509 0.90 ALDH1A1 (0.49) ALDH1A1MITFHTTHPGD
SCHEMBL9897513 0.90 ALDH1A1 (0.49) ALDH1A1MITFHTTHPGD
SCHEMBL9899508 0.89 PTGES (0.44) ALDH1A1HCAR3MITFCDC25BPOLB
SCHEMBL9899506 0.89 PTGES (0.44) ALDH1A1HCAR3MITFCDC25BPOLB
SCHEMBL27924938 0.85 ALDH1A1 (0.40) ALDH1A1HCAR3MITFCDC25BPOLB
SCHEMBL9898930 0.84 ALDH1A1 (0.45) ALDH1A1MITFPOLBL3MBTL1HPGD
SCHEMBL9898933 0.84 ALDH1A1 (0.45) ALDH1A1MITFPOLBL3MBTL1HPGD
SCHEMBL9899352 0.84 PTGES (0.43) ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012076673-A1 6-AMINO-2-PHENYLAMINO-1H-BENZIMIDAZOLE-5-CARBOXAMIDE- DERIVATIVES AND THEIR USE AS MICROSOMAL PROSTAGLANDIN E2 SYNTHASE-1 INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-06-14 WO disclosed